BDBM50585044 CHEMBL5088392
SMILES [H][C@@]12[C@@H](C)OC(=O)[C@@]11CN(C[C@H]1[C@H](C)[C@@H](C)[C@@H]2\C=C\c1ccc(cn1)-c1ccccc1C#N)C(=O)NCC
InChI Key InChIKey=UAELFEWPCXTKFL-IDKUMADTSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50585044
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human PAR-1 expressed in HEK293 cells assessed as reduction in TRAP induced calcium signal at 3 uM by FLIPR analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of [35S]MK-499 binding to hERG expressed in HEK293 cells at 60 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of [35S]MK-499 binding to hERG expressed in HEK293 cellsMore data for this Ligand-Target Pair