BDBM523849 US11136320, Compound 8

SMILES CO[C@@H]1CCN(Cc2cc3CCCN(C(=O)Nc4cc(NCCSC)c(cn4)C#N)c3nc2OC)C1=O

InChI Key InChIKey=ZKGQVQGIVCBSTA-HXUWFJFHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 523849   

TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523849(US11136320, Compound 8)
Affinity DataIC50:  0.420nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent