BDBM536813 5-(8-(5-acetyl-1-(tetrahydro-2H-pyran-4-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-4-fluoroisoquinolin-3-yl)-N-methylpicolinamide::US11247989, Example 24
SMILES CNC(=O)c1ccc(cn1)-c1ncc2c(cccc2c1F)-c1nn(C2CCOCC2)c2CCN(Cc12)C(C)=O
InChI Key InChIKey=TUVOZXGYQPNWGN-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 536813
Affinity DataIC50: 2.05nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair