BDBM602184 US11643436, Compound TM-7

SMILES CC(C)C[C@@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1)C(=O)N[C@H](CCCCN)C(=O)N1CCC2(CC(C2)B(O)O)CC1

InChI Key InChIKey=BPHFEGXYOHHBCT-XEXPGFJZSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 602184   

TargetKappa-type opioid receptor(Homo sapiens (Human))
Chengdu Sintanovo Biotechnology

US Patent
LigandPNGBDBM602184(US11643436, Compound TM-7)
Affinity DataEC50:  0.00900nMAssay Description:Forskolin can stimulate the release of cAMP from HEK293 cells with high expression of human κ (or μ, or δ)-opioid receptors. The κ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Chengdu Sintanovo Biotechnology

US Patent
LigandPNGBDBM602184(US11643436, Compound TM-7)
Affinity DataEC50: >1.00E+4nMAssay Description:Forskolin can stimulate the release of cAMP from HEK293 cells with high expression of human κ (or μ, or δ)-opioid receptors. The κ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDelta-type opioid receptor(Homo sapiens (Human))
Chengdu Sintanovo Biotechnology

US Patent
LigandPNGBDBM602184(US11643436, Compound TM-7)
Affinity DataEC50: >1.00E+4nMAssay Description:Forskolin can stimulate the release of cAMP from HEK293 cells with high expression of human κ (or μ, or δ)-opioid receptors. The κ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent