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Found 25 with Last Name = 'eleutheriades' and Initial = 'a'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382166(CHEMBL2023825)
Affinity DataIC50:  0.270nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401861(CHEMBL2204672)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382169(CHEMBL2023824)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382165(CHEMBL2023823)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401862(CHEMBL2204668)
Affinity DataIC50:  5.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401857(CHEMBL2204679)
Affinity DataIC50:  12.3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382168(CHEMBL2023827)
Affinity DataIC50:  12.4nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401859(CHEMBL2204677)
Affinity DataIC50:  36.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401858(CHEMBL2204678)
Affinity DataIC50:  42nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50401860(CHEMBL2204675)
Affinity DataIC50:  48.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382167(CHEMBL2023826)
Affinity DataIC50:  63.3nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50382164(CHEMBL2023828)
Affinity DataIC50: >100nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423058(CHEMBL244471)
Affinity DataIC50:  282nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423056(CHEMBL243002)
Affinity DataIC50:  1.18E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423059(CHEMBL244472)
Affinity DataIC50:  1.41E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423057(CHEMBL242573)
Affinity DataIC50:  1.51E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423062(CHEMBL242786)
Affinity DataIC50:  1.59E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423063(CHEMBL396501)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423061(CHEMBL243003)
Affinity DataIC50:  2.04E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423055(CHEMBL244957)
Affinity DataIC50:  2.19E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM85065(CAS_117946-91-5 | Luzindole | NSC_122162)
Affinity DataIC50:  2.46E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423064(CHEMBL244263)
Affinity DataIC50:  4.68E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423060(CHEMBL241928)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50423065(CHEMBL242806)
Affinity DataIC50:  6.17E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Xenopus)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50411361(CHEMBL396991)
Affinity DataIC50:  1.00E+5nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed