TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 12.3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 12.4nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 36.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 48.1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in human Jurkat cell membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 63.3nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Displacement of [3H](+)pentazocine from sigma-1 receptor expressed in human Jurkat cell membranes after 2 hrs by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.46E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.68E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.17E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair