TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of serum-stimulated proliferation of mouse ERBB2 transfected NIH3T3 cell line after 24 hrsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 204nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 294nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 335nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 482nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 508nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of serum-stimulated proliferation of mouse ERBB2 transfected NIH3T3 cell line after 24 hrsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 676nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of serum-stimulated proliferation of mouse ERBB2 transfected NIH3T3 cell line after 24 hrsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of serum-stimulated proliferation of mouse ERBB2 transfected NIH3T3 cell line after 24 hrsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 903nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EGFR tyrosine kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair