TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of radioligand from human recombinant adenosine A2A receptor at 21 degC after 90 mins by cell-based microplate scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair