Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]Oxytocin from human OXTR expressed in CHO cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]Oxytocin from human OXTR expressed in CHO cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement of [3H]-AVP from human V1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Displacement of [3H]-AVP from human V1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1b receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1b receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1b receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-AVP from human V1b receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Displacement of [3H]-AVP from human V1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.70E+3nMAssay Description:Displacement of [3H]-AVP from human V1A receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.60E+3nMAssay Description:Displacement of [3H]-AVP from human V1b receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human BChE after 30 mins by microplate reader methodMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human BChE after 30 mins by microplate reader methodMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 61.2nMAssay Description:Inhibition of human BChE after 30 mins by microplate reader methodMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:The 1321N1 cells stably expressing human P2X4 receptor were seeded on a 96-well plate, cultured under the conditions of 37° C. and 5% CO2 for 24 hour...More data for this Ligand-Target Pair