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Found 79 with Last Name = 'crist' and Initial = 'm'
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089280(CHEMBL437655 | JMV 1535)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089284(CHEMBL265856 | JMV 1803)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089285(CHEMBL415110 | JMV 1799)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089281(CHEMBL386480 | JMV 1802)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089291(CHEMBL415021 | JMV 1813)
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089278(CHEMBL411016 | JMV 1801)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089279(CHEMBL406013 | JMV 1719)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089286(CHEMBL407022 | JMV 1693)
Affinity DataKi:  127nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408922(CHEMBL2115179)
Affinity DataKi:  225nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089288(Bombesin analogues | CHEMBL415022)
Affinity DataKi:  300nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089292(Bombesin analogues | CHEMBL439440)
Affinity DataKi:  500nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089290(Bombesin analogues | CHEMBL413938)
Affinity DataKi:  650nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089293(Bombesin analogues | CHEMBL407481)
Affinity DataKi:  2.25E+3nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089287(Bombesin analogues | CHEMBL384242)
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089289(Bombesin analogues | CHEMBL384241)
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299583((S)-N-(3-bromophenyl)-N'-cyano-2-methyl-4-(5-methy...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of LIMK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299619((S)-3-(N'-cyano-2-methyl-4-(5-methyl-7H-pyrrolo[2,...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299583((S)-N-(3-bromophenyl)-N'-cyano-2-methyl-4-(5-methy...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299616((S)-N-(3-tert-butylphenyl)-N'-cyano-2-methyl-4-(5-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299607((S)-N-(3-bromophenyl)-4-(5-chloro-7H-pyrrolo[2,3-d...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299586((S)-3-(2-methyl-4-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299615((S)-N'-cyano-N-(3-cyanophenyl)-2-methyl-4-(5-methy...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299584((S)-N-(3-bromo-4-fluorophenyl)-N'-cyano-2-methyl-4...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299611((S)-N-(3-chlorophenyl)-N'-cyano-2-methyl-4-(5-meth...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299623((S)-N'-cyano-N-(3-(N-isopropylsulfamoyl)phenyl)-2-...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299613((S)-N'-cyano-N-(3-fluorophenyl)-2-methyl-4-(5-meth...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299614((S)-N'-cyano-2-methyl-4-(5-methyl-7H-pyrrolo[2,3-d...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Algarve

Curated by ChEMBL
LigandPNGBDBM50243232(CHEMBL486232 | GNF-PF-5434 | N-((S)-4-methyl-1-oxo...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299612((S)-N-(3-chlorophenyl)-2-methyl-4-(5-methyl-7H-pyr...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299624((S)-N'-cyano-N-(3-(N-(2-hydroxyethyl)sulfamoyl)phe...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299620((S)-N-(3-(2-hydroxyethylcarbamoyl)phenyl)-2-methyl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299621((S)-N-(3-(1,3-dihydroxypropan-2-ylcarbamoyl)phenyl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299586((S)-3-(2-methyl-4-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of LIMK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299585((S)-N-(3-bromo-4-fluorophenyl)-2-methyl-4-(5-methy...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299622((S)-3-(N'-cyano-2-methyl-4-(5-methyl-7H-pyrrolo[2,...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299617((S)-3-(N'-cyano-2-methyl-4-(5-methyl-7H-pyrrolo[2,...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299584((S)-N-(3-bromo-4-fluorophenyl)-N'-cyano-2-methyl-4...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of LIMK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299599((S)-N-(3-bromophenyl)-2-methyl-4-(5-methyl-7H-pyrr...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299602(CHEMBL570586 | Trans-N-(3-bromophenyl)-N'-cyano-2,...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299601((S)-N-(3-bromophenyl)-N'-cyano-2-isopropyl-4-(5-me...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299608((S)-N-(3-bromophenyl)-N'-cyano-2-methyl-4-(6-methy...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299618((S)-N-(3-(isopropylcarbamoyl)phenyl)-2-methyl-4-(5...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 1(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299585((S)-N-(3-bromo-4-fluorophenyl)-2-methyl-4-(5-methy...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of LIMK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299610((S)-N-(3-bromophenyl)-2-methyl-4-(5-methyl-7H-pyrr...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299606((+/-)-N-(3-bromophenyl)-N'-cyano-2-methyl-4-(7H-py...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299598(CHEMBL568484 | N-(3-bromophenyl)-N'-cyano-4-(5-met...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLIM domain kinase 2(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299604(CHEMBL584968 | N-(3-bromophenyl)-3-(5-methyl-7H-py...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant LIMK2 expressed in baculovirus-Sf9 system by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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