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Found 41 with Last Name = 'ganapathy' and Initial = 'me'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM85392(CAS_131443 | NSC_131443 | PPAP, (-))
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataKi:  8.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM94507(2-[2-(diethylamino)ethoxy]ethyl 1-phenylcyclopenta...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM85391(CAS_85976-54-1 | NSC_149136 | PPP, (+))
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM81982(CAS_97-39-2 | DITOLYLGUANIDINE | DTG | Di-o-tolylg...)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  353nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medical College of Georgia

Curated by PDSP Ki Database
LigandPNGBDBM50003560(4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.0...)
Affinity DataKi:  521nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350467(BL-S578 | CEFADROXIL | Cefadrops)
Affinity DataKi:  2.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Chephalexin uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350467(BL-S578 | CEFADROXIL | Cefadrops)
Affinity DataKi:  2.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  1.40E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350474(CICLACILLIN | CYCLACILLIN)
Affinity DataKi:  3.68E+4nMAssay Description:TP_TRANSPORTER: inhibition of Chephalexin uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350474(CICLACILLIN | CYCLACILLIN)
Affinity DataKi:  3.91E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  4.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM81945(CAS_39484 | CHEMBL105891 | CHEMBL108926 | CHEMBL27...)
Affinity DataKi:  5.40E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50188516(2-(2-amino-N-methylacetamido)acetic acid | CHEMBL1...)
Affinity DataKi:  6.40E+4nMAssay Description:TP_TRANSPORTER: inhibition of Cephalexin uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50139896((6R,7R)-7-((R)-2-Amino-2-phenyl-acetylamino)-3-met...)
Affinity DataKi:  6.82E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(7-(2-(2-amino-4-thiazolyl)-4-carboxy-2-butenoylami...)
Affinity DataKi:  9.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Rattus norvegicus)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  1.70E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50225285(CHEBI:3757 | Catapres | Catapres-Tts-1 | Catapres-...)
Affinity DataKi:  3.73E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(7-(2-(2-amino-4-thiazolyl)-4-carboxy-2-butenoylami...)
Affinity DataKi:  3.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  3.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  4.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(7-(2-(2-amino-4-thiazolyl)-4-carboxy-2-butenoylami...)
Affinity DataKi:  7.10E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM39344(4-amino-N-[2-(diethylamino)ethyl]benzamide;hydroch...)
Affinity DataKi:  7.38E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  7.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(7-(2-(2-amino-4-thiazolyl)-4-carboxy-2-butenoylami...)
Affinity DataKi:  8.70E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  1.37E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataKi:  6.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350467(BL-S578 | CEFADROXIL | Cefadrops)
Affinity DataIC50:  6.60E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 50 uM) in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50103624(40602 | CHEBI:3537 | Cefaloridine | Cephaloridine ...)
Affinity DataIC50:  2.30E+5nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350474(CICLACILLIN | CYCLACILLIN)
Affinity DataIC50:  3.50E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 25 uM) in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350474(CICLACILLIN | CYCLACILLIN)
Affinity DataIC50:  6.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350474(CICLACILLIN | CYCLACILLIN)
Affinity DataIC50:  6.10E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 50 uM) in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350467(BL-S578 | CEFADROXIL | Cefadrops)
Affinity DataIC50:  8.70E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 25 uM) in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350470(CEFEPIME | Maxipime)
Affinity DataIC50:  1.70E+6nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataIC50:  3.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50350467(BL-S578 | CEFADROXIL | Cefadrops)
Affinity DataIC50:  5.40E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataIC50:  1.00E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 15 member 2(Rattus norvegicus)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50248190(CHEBI:3485 | CI-983 | Cefdinir | Cefzon | FK-482 |...)
Affinity DataIC50:  1.00E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 5(Homo sapiens)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50485614(Cefoselis)
Affinity DataIC50:  6.40E+7nMAssay Description:TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed