Found 7 Enz. Inhib. hit(s) with Target = 'Solute carrier family 15 member 1' and Ligand = 'BDBM50350467'
Affinity DataKi: 1.45E+6nMAssay Description:TP_TRANSPORTER: inhibition of Cefixim uptake in Caco-2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 15 member 1(Rattus norvegicus)
Kyoto University Hospital
Curated by ChEMBL
Kyoto University Hospital
Curated by ChEMBL
Affinity DataKi: 2.17E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+6nMAssay Description:Binding affinity against membrane transport protein PEPT1 in human Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.10E+6nMAssay Description:TP_TRANSPORTER: inhibition of VACV uptake in PEPT1-expressing CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 25 uM) in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair