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Found 26 with Last Name = 'gkeka' and Initial = 'p'
TargetCarboxypeptidase B2(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547476(CHEMBL4782260)
Affinity DataIC50:  10nMAssay Description:Inhibition of TAFIalpha in human plasma incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM173926(US9688645, 7-1)
Affinity DataIC50:  22nMAssay Description:Inhibition of TAFIalpha in human plasma incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547477(CHEMBL4764267)
Affinity DataIC50:  42nMAssay Description:Inhibition of TAFIalpha in human plasma incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547478(CHEMBL4743386)
Affinity DataIC50:  52nMAssay Description:Inhibition of TAFIalpha in human plasma incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547471(CHEMBL4762061)
Affinity DataEC50:  0.194nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547472(CHEMBL4761047)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547473(CHEMBL4757675)
Affinity DataEC50:  0nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547474(CHEMBL4741348)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547475(CHEMBL4745985)
Affinity DataEC50:  0.0480nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50266674(CHEMBL4098061)
Affinity DataEC50:  0.0180nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547466(CHEMBL4751319)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547467(CHEMBL4755815)
Affinity DataEC50:  0.0540nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547468(CHEMBL4758415)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547469(CHEMBL4756489)
Affinity DataEC50:  8.43nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547470(CHEMBL4745235)
Affinity DataEC50:  0.122nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547471(CHEMBL4762061)
Affinity DataEC50:  0.578nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547472(CHEMBL4761047)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547473(CHEMBL4757675)
Affinity DataEC50:  0.369nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547474(CHEMBL4741348)
Affinity DataEC50:  0.00200nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547475(CHEMBL4745985)
Affinity DataEC50:  0.119nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50266674(CHEMBL4098061)
Affinity DataEC50:  0.0290nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547470(CHEMBL4745235)
Affinity DataEC50:  0.0750nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547469(CHEMBL4756489)
Affinity DataEC50:  0.00100nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547468(CHEMBL4758415)
Affinity DataEC50:  0.00600nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547466(CHEMBL4751319)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Schrodinger

Curated by ChEMBL
LigandPNGBDBM50547467(CHEMBL4755815)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human GLP-1 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed