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Found 100 with Last Name = 'cheruvallath' and Initial = 'zs'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212260(CHEMBL3954836)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212261(CHEMBL3946139)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212254(CHEMBL3975466)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212256(CHEMBL3966978)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212280(CHEMBL3962015)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212284(CHEMBL3925645)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212262(CHEMBL3937245)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212263(CHEMBL3928256)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212257(CHEMBL3943495)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212278(CHEMBL3934521)
Affinity DataIC50:  32nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212259(CHEMBL3953259)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212265(CHEMBL3890544)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212285(CHEMBL3891901)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212255(CHEMBL3960900)
Affinity DataIC50:  398nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212279(CHEMBL3955870)
Affinity DataIC50:  794nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431731(CHEMBL2346751)
Affinity DataEC50:  160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431732(CHEMBL2346752)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431733(CHEMBL2346756)
Affinity DataEC50:  630nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431734(CHEMBL2346755)
Affinity DataEC50:  500nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431735(CHEMBL2346754)
Affinity DataEC50:  160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431736(CHEMBL2346753)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431737(CHEMBL2346757)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431738(CHEMBL2346758)
Affinity DataEC50:  200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431739(CHEMBL2346759)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431740(CHEMBL2346760)
Affinity DataEC50:  790nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431741(CHEMBL2346761)
Affinity DataEC50:  79nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431742(CHEMBL2346762)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431743(CHEMBL2346763)
Affinity DataEC50:  6.30E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431744(CHEMBL2346764)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431745(CHEMBL2346875)
Affinity DataEC50:  400nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431746(CHEMBL2346877)
Affinity DataEC50:  160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431747(CHEMBL2346876)
Affinity DataEC50:  250nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431748(CHEMBL2346667)
Affinity DataEC50:  200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431749(CHEMBL2346879)
Affinity DataEC50:  200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431750(CHEMBL2346878)
Affinity DataEC50:  310nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431751(CHEMBL2346880)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431752(CHEMBL2346881)
Affinity DataEC50:  790nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431753(CHEMBL2346882)
Affinity DataEC50:  63nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431754(CHEMBL2346883)
Affinity DataEC50:  250nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431755(CHEMBL2346884)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431756(CHEMBL2346885)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431757(CHEMBL2346886)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431758(CHEMBL2346887)
Affinity DataEC50:  630nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431759(CHEMBL2346888)
Affinity DataEC50:  400nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431760(CHEMBL2346892)
Affinity DataEC50:  310nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431761(CHEMBL2346891)
Affinity DataEC50:  79nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50431762(CHEMBL2346890)
Affinity DataEC50:  2.50E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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