TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 790nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 6.30E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 790nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Activation of glucokinase (unknown origin)More data for this Ligand-Target Pair