Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 5' and Ligand = 'BDBM50212282'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin) using biotin-MBP as substrate after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ASK1 catalytic domain (654 to 971 residues) expressed in baculovirus infected sf21 cells using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed