Affinity DataKi: 0.0500nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of Epidermal growth factor receptor from human A431 cell membranesMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to HIV-1 protease assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase K103NMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase G190AMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand Info
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase K103NMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against HIV-1 Y188L reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase G190AMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against HIV-1 Y188L reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase G190AMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase K103NMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:The COX activity was assayed colorimetrically by monitoring the appearance of oxidized N,N,N',N'-tetramethyl-pphenylenediamine (TMPD) at 590 ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase P236LMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase V106AMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Alwar Pharmacy College
Curated by ChEMBL
Alwar Pharmacy College
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 225nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair