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Found 741 with Last Name = 'avery' and Initial = 'm'
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  0.0140nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  0.0160nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  0.0190nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.0280nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  0.0350nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  0.0380nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  0.0530nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50550643(CHEMBL4749207)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to human 20S constitutive proteasome beta 5 subunit assessed as equilibrium constant using fluorogenic peptide Ac-WLA-AMC as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  0.154nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM420298(CVD-0006356 | PF-00835231 | PF-0835231 | US1152494...)
Affinity DataKi:  0.270nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
Ligand InfoPurchasePDB
In DepthDetails PDB3D3D Structure (crystal)
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.700nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.800nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM496902(CVD-0018409 | PF-07321332 | US11351149, Example 13...)
Affinity DataKi:  3.11nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  4nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  5.5nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM496900(science.abl4784, 4)
Affinity DataKi:  7.93nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM496901(science.abl4784, 5)
Affinity DataKi:  12nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303975(3'-(4-(2-(1H-Tetrazol-5-yl)ethyl)benzyl)-1,7'-dime...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  15nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  23nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM496896(US11312704, Compound 101 | US11351149, Example 49 ...)
Affinity DataKi:  28nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  41nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  75nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  86nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  113nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50504220(CHEMBL4454497)
Affinity DataKi:  200nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

LigandPNGBDBM496897(science.abl4784, 3)
Affinity DataKi:  230nMAssay Description:The respective human coronavirus Mpro in assay buffer (20 mM Tris-HCl, pH 7.3, 100 mM NaCl, 1 mM EDTA, 5 mM TCEP) and 0.1% BSA was added to assay-rea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAminopeptidase N(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50518449(CHEMBL4435950)
Affinity DataKi:  300nMAssay Description:Inhibition of human APN expressed in HEK293 cells preincubated for 20 mins followed by L-leucine-7-amido-4-methylcoumarin addition by fluorescence as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi:  390nMAssay Description:Binding affinity to 5HT2B receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50504218(CHEMBL4437088)
Affinity DataKi:  400nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi:  464nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
The University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50550643(CHEMBL4749207)
Affinity DataKi:  487nMAssay Description:Binding affinity to human 20S constitutive proteasome beta 2 subunit assessed as equilibrium constant using fluorogenic peptide Ac-WLR-AMC as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi:  560nMAssay Description:Binding affinity to sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
The Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50504225(CHEMBL4546549)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303976(3'-(2-(4-(2-(1H-Tetrazol-5-yl)ethyl)phenoxy)ethyl)...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303977(3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'-biben...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303979(CHEMBL571763 | Ethyl 3-(4-(2-(1,7'-Dimethyl-2'-pro...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303978(1-(4-(2-(1H-tetrazol-5-yl)ethyl)benzyl)-4-methyl-2...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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