Affinity DataKi: 0.230nM ΔG°: -55.0kJ/molepH: 7.5 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Competitive reversible inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
University Of Liverpool
Curated by ChEMBL
University Of Liverpool
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Inhibition of Cyclophilin D (unknown origin) activity in absence of detergentMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/molepH: 7.5 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:The compound was tested for its inhibitory activity against IL-1 beta converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:The compound was tested for its inhibitory activity against IL-1 beta converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
University Of Liverpool
Curated by ChEMBL
University Of Liverpool
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Inhibition of Cyclophilin D (unknown origin) activity preincubated for 15 mins followed Suc-AAPF-pNA substrate addition by chymotrypsin coupled based...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:The compound was tested for its inhibitory activity against IL-1 beta converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Tested for inhibition of cysteine proteinase IL-1 beta converting enzyme (ICE)More data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 133nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Compound was tested for its inhibition against Caspase-8More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity determined against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:The compound was tested for its inhibitory activity against IL-1 beta converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity of the compound was determined against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
University Of Liverpool
Curated by ChEMBL
University Of Liverpool
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:Inhibition of Cyclophilin D (unknown origin) activity preincubated for 15 mins followed Suc-AAPF-pNA substrate addition by chymotrypsin coupled based...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity of the compound was determined against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for Potassium channel HERG Kv11.1More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
University Of Liverpool
Curated by ChEMBL
University Of Liverpool
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of Cyclophilin D (unknown origin) activity preincubated for 15 mins followed Suc-AAPF-pNA substrate addition by chymotrypsin coupled based...More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair