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Found 44 with Last Name = 'canettieri' and Initial = 'g'
TargetL-lactate dehydrogenase B chain(Mus musculus (Mouse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of mouse LDHB using sodium pyruvate as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human LDHA using sodium pyruvate as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50592886(CHEMBL5199516)
Affinity DataKi:  5.46E+3nMAssay Description:Inhibition of LDHA in human liver using pyruvate as substrate incubated for 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50592886(CHEMBL5199516)
Affinity DataKi:  1.51E+4nMAssay Description:Inhibition of LDHB in human heart using pyruvate as substrate incubated for 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50144744(Sodium Oxamate)
Affinity DataKi:  1.36E+5nMAssay Description:Inhibition of human LDHA using sodium pyruvate as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50592885(CHEMBL5206296)
Affinity DataIC50:  12nMAssay Description:Inhibition of LDHA in human Med1 cells using pyruvate as substrate incubated 10 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509994(CHEMBL4449346)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509991(CHEMBL4539177)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509988(CHEMBL4584542)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509997(CHEMBL4527356)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509989(CHEMBL4536754)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509991(CHEMBL4539177)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50144744(Sodium Oxamate)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of LDHA in human Med1 cells using pyruvate as substrate incubated 10 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50510000(CHEMBL4456805)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509999(CHEMBL2363137)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509989(CHEMBL4536754)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509993(CHEMBL4473926)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509995(CHEMBL4455336)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509996(CHEMBL4546428)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM35617(5-chloroindolecarboxamide, 2a)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509990(CHEMBL4436448)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509985(CHEMBL4588868)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509986(CHEMBL4453345)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509992(CHEMBL4439563)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509987(CHEMBL4454568)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509988(CHEMBL4584542)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509994(CHEMBL4449346)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509997(CHEMBL4527356)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of NHERF1 in human SW620 cells expressing NHERF1 assessed as inhibition cell growth incubated for 72 hrs by MTT assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509991(CHEMBL4539177)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509998(CHEMBL4458535)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509996(CHEMBL4546428)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM35617(5-chloroindolecarboxamide, 2a)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509995(CHEMBL4455336)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509993(CHEMBL4473926)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509990(CHEMBL4436448)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509985(CHEMBL4588868)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509987(CHEMBL4454568)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509986(CHEMBL4453345)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509992(CHEMBL4439563)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509989(CHEMBL4536754)
Affinity DataIC50:  7.40E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509988(CHEMBL4584542)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509994(CHEMBL4449346)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509997(CHEMBL4527356)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50509998(CHEMBL4458535)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of NHERF1 in human Ls174T cells stably transfected with Dox-inducible shRNA for beta-catenin (Ls174Tsh-beta-Cat) assessed as inhibition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed