Affinity DataIC50: 8nMAssay Description:Inhibition of Zea mays (maize) chloroplastic ACCase using acetyl-coA as substrate assessed as inhibition of [14C]NaHCO3 incorporation into malonyl-co...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Zea mays (maize) cytosolic ACCase using acetyl-coA as substrate assessed as inhibition of [14C]NaHCO3 incorporation into malonyl-coA in...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Zea mays (maize) chloroplastic ACCase using acetyl-coA as substrate assessed as inhibition of [14C]NaHCO3 incorporation into malonyl-co...More data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 4.84E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 6.93E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 8.03E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 8.61E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Zea mays (maize) cytosolic ACCase using acetyl-coA as substrate assessed as inhibition of [14C]NaHCO3 incorporation into malonyl-coA in...More data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven
Curated by ChEMBL
Katholieke Universiteit Leuven
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 5.19E+4nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 5.73E+4nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 7.51E+4nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >8.79E+4nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >9.04E+4nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 9.28E+4nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.08E+5nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.13E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.18E+5nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.18E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.19E+5nMAssay Description:Inhibition of Mycobacterium smegmatis MC2 DNA gyrase GyrB ATPase supercoiling activityMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Mycobacterium smegmatis)
Birla Institute Of Technology And Science
Curated by ChEMBL
Birla Institute Of Technology And Science
Curated by ChEMBL
Affinity DataIC50: >1.32E+5nMAssay Description:Inhibition of Mycobacterium smegmatis DNA gyraseMore data for this Ligand-Target Pair