Affinity DataKi: 0.300nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity toward 5-HT2B receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity toward 5-HT2C receptor evaluated by displacement of [3H]-5-HT radioligand More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity toward 5-HT2A receptor evaluated by displacement of [125I]-DOI radioligand More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair