Affinity DataKi: 0.600nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [125I]peptideYY from NPY1 receptor in human SK-N-MC cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.66E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 4.79E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 5.78E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 7.18E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 9.50E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.29E+6nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair
TargetPresenilin-1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of gamma secretase-mediated beta-APP cleavage in human H4 cells assessed by measuring Abeta40 production by ELISAMore data for this Ligand-Target Pair