TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Brookhaven National Laboratory
Curated by ChEMBL
Brookhaven National Laboratory
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]epibatidine from alpha-4-beta-2 ACHRMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BTK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of Ron (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of c-MET (unknown origin) using peptide as substrate incubated for 1 hr by mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of Tyro3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >5nMAssay Description:Inhibition of JAK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of BTK (unknown origin) assessed as reduction in TNF productionMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of MEK1 in mouse C2C12 by ERK2 phosphorylation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
College Of Pharmacy Of Liaoning University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of ITK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of ErbB4/HER4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair