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Found 384 with Last Name = 'ding' and Initial = 's'
TargetUrotensin-2 receptor(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86516(ETPDCFWKYCV | Human U-II | L-Ala-Gly-L-Thr-L-Ala-L...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Actelion Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86516(ETPDCFWKYCV | Human U-II | L-Ala-Gly-L-Thr-L-Ala-L...)
Affinity DataKi:  6.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Brookhaven National Laboratory

Curated by ChEMBL
LigandPNGBDBM50177228(7-methyl-2-exo-(3'-iodo-5'-pyridinyl)-7-azabicyclo...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]epibatidine from alpha-4-beta-2 ACHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Actelion Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50302272(1-(2-(4-benzyl-4-hydroxypiperidin-1-yl)ethyl)-3-(2...)
Affinity DataKi:  1.48E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM1774(US10894048, Ref. Ex Comp. 1 | US8476284, 13)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of BTK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50551837(CHEMBL4753082)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369720(CHEMBL3979355)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50551837(CHEMBL4753082)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of Ron (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM36516(4-(tert-Butyl)-N-(2-methyl-3-(4-methyl-6-((4-(morp...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369721(CHEMBL3702836)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369718(CHEMBL4172284)
Affinity DataIC50:  2nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455107(CHEMBL4212167)
Affinity DataIC50:  2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455106(CHEMBL4216095)
Affinity DataIC50:  2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455115(CHEMBL4202932)
Affinity DataIC50:  2nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369722(CHEMBL4175428)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024529(CHEMBL3330482)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50175583(ACP-196 | Acalabrutinib | US10239883, Example 6 | ...)
Affinity DataIC50:  3nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455105(CHEMBL4218384)
Affinity DataIC50:  3nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024356(CHEMBL3330442)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50551837(CHEMBL4753082)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136890(CHEMBL152208 | [2-Chloro-4-(4-fluoro-2-methyl-phen...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50388189(CHEMBL2057918)
Affinity DataIC50:  4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369723(CHEMBL4167139)
Affinity DataIC50:  4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50:  4nMAssay Description:Inhibition of c-MET (unknown origin) using peptide as substrate incubated for 1 hr by mobility shift assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50551837(CHEMBL4753082)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of Tyro3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024538(CHEMBL3330490)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024530(CHEMBL3330483)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
LigandPNGBDBM50369720(CHEMBL3979355)
Affinity DataIC50: >5nMAssay Description:Inhibition of JAK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136887(CHEMBL356455 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024536(CHEMBL3330493)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369722(CHEMBL4175428)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369719(CHEMBL4162057)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455114(CHEMBL4207862)
Affinity DataIC50:  6nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50024540(CHEMBL3330491)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50388189(CHEMBL2057918)
Affinity DataIC50:  7nMAssay Description:Inhibition of BTK (unknown origin) assessed as reduction in TNF productionMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136897((2-Chloro-4-phenylamino-phenyl)-o-tolyl-methanone ...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455112(CHEMBL4215964)
Affinity DataIC50:  7nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50170831(CHEMBL188343 | N*6*-Cyclohexyl-N*2*-(4-morpholin-4...)
Affinity DataIC50:  8nMAssay Description:Inhibition of MEK1 in mouse C2C12 by ERK2 phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50012060(CHEMBL3263640)
Affinity DataIC50:  8nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus 14)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50455113(CHEMBL4212963)
Affinity DataIC50:  8nMAssay Description:Inhibition of Human rhinovirus serotype 14 3C protease preincubated for 1 hr followed by Cys(PT14M)-Ala-Ile-Phe-Gln'Gly-Pro-Asp-Phe(4-NH2)-OH substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM7840(RIVAROXABAN | US8822458, 44 | US8822458, 97)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of human factor 10a using N-Z-D-Arg-Gly-Arg-pNA, S-2765 chromogenic substrateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136886(CHEMBL152767 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
College Of Pharmacy Of Liaoning University

Curated by ChEMBL
LigandPNGBDBM50598528(CHEMBL5201846)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM1774(US10894048, Ref. Ex Comp. 1 | US8476284, 13)
Affinity DataIC50:  11nMAssay Description:Inhibition of ITK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Shaanxi University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50369720(CHEMBL3979355)
Affinity DataIC50:  11nMAssay Description:Inhibition of ErbB4/HER4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136884((2-Chloro-4-o-tolylamino-phenyl)-o-tolyl-methanone...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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