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Found 123 with Last Name = 'foleno' and Initial = 'bd'
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against class A Beta-lactamase TEM isolated from Enterobacter coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092284(5-[(E)-3-(5-Nitro-furan-2-yl)-prop-2-en-(Z)-yliden...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092281(3-[4-Oxo-2-thioxo-thiazolidin-(5E)-ylidene]-1,3-di...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471725(CHEMBL327734)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215968(CHEMBL57324)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50063753(CHEMBL12131 | Closantel | N-(5-chloro-4-((4-chloro...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092283(5-[(E)-3-(4-Nitro-phenyl)-prop-2-en-(Z)-ylidene]-2...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471718(CHEMBL98026)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215967(CHEMBL56579)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218645(CHEMBL288462)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218644(CHEMBL416972)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215985(CHEMBL57037)
Affinity DataIC50:  8.00E+3nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092286(5-[(E)-3-(4-Dimethylamino-phenyl)-prop-2-en-(Z)-yl...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092281(3-[4-Oxo-2-thioxo-thiazolidin-(5E)-ylidene]-1,3-di...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory activity against class A Beta-lactamase TEM isolated from Enterobacter coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471730(CHEMBL101786)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation initiation phosphotransferase F/kinase A(Bacillus subtilis (strain 168))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215963(CHEMBL57687)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471728(CHEMBL100719)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092279(5-[3-Phenyl-prop-(Z)-ylidene]-2-thioxo-thiazolidin...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218648(CHEMBL290098)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218640(CHEMBL38683)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218643(CHEMBL39634)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218655(CHEMBL38914)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218647(CHEMBL38867)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215976(CHEMBL58536)
Affinity DataIC50:  1.60E+4nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218659(CHEMBL43691)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471723(CHEMBL98273)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50065970(CHEMBL57656 | N-(3,4-Dichloro-phenyl)-2-hydroxy-3,...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50065970(CHEMBL57656 | N-(3,4-Dichloro-phenyl)-2-hydroxy-3,...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215978(CHEMBL58439)
Affinity DataIC50:  2.40E+4nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218653(CHEMBL39178)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471716(CHEMBL431272)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50100895(2-(4-(4-carbamimidoylphenoxy)phenyl)-1H-indole-6-c...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of KinA/Sp0F system two component system (TCS) from Bacillus subtilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092279(5-[3-Phenyl-prop-(Z)-ylidene]-2-thioxo-thiazolidin...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity against class A Beta-lactamase TEM isolated from Enterobacter coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215974(3,3'',4'',5-tetrachlorosalicylanilide | 3,3',4',5-...)
Affinity DataIC50:  3.70E+4nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218651(CHEMBL39490)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of KinA/Sp0F two component system (TCS) from Bacillus subtilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092268(5-(4-nitrobenzylidene)-2-thioxothiazolidin-4-one |...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218656(CHEMBL39040)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215977(CHEMBL58560)
Affinity DataIC50:  4.40E+4nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215974(3,3'',4'',5-tetrachlorosalicylanilide | 3,3',4',5-...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of histidine protein kinase (KinA) phosphorylation in the presence of response regulator (Spo0F)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215974(3,3'',4'',5-tetrachlorosalicylanilide | 3,3',4',5-...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218646(CHEMBL290549)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092269(5-[(E)-3-(5-Nitro-furan-2-yl)-prop-2-en-(Z)-yliden...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against class A Beta-lactamase TEM isolated from Enterobacter coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471712(CHEMBL319252)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092269(5-[(E)-3-(5-Nitro-furan-2-yl)-prop-2-en-(Z)-yliden...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092282(5-[(E)-3-Furan-2-yl-prop-2-en-(Z)-ylidene]-2-thiox...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218654(CHEMBL40096)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50216089(CHEMBL441791)
Affinity DataIC50:  6.70E+4nMAssay Description:Ability to inhibit autophosphorylation of KinA/Sp0F assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50471719(CHEMBL100688)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of autophosphorylation of the two-component signal transduction system kinase was measured using the KinA/Spo0F regulatory system of Bacil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSporulation kinase A(Bacillus subtilis (strain 168))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50218649(CHEMBL417892)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of KinA/Sp0F system two component (TCS) from Bacillus subtilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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