Affinity DataKi: 0.0940nMAssay Description:Binding affinity for human fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity for rat fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]CP-55940 binding to human cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: 9.10nMAssay Description:Binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for human cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: 96nMAssay Description:Apparent binding affinity for fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Noncompetitive inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of FAAH-mediated [3H]AEA hydrolysis in rat brain homogenate by time-dependent studiesMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of FAAH-mediated [3H]AEA hydrolysis in rat brain homogenate by time-dependent studiesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: 250nMAssay Description:Binding affinity for cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Competitive inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: 442nMAssay Description:Inhibition of [3H]CP-55940 binding to human cannabinoid receptor 2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: 800nMAssay Description:Binding affinity for Cannabinoid receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D
Curated by PDSP Ki Database
Astrazeneca R&D
Curated by PDSP Ki Database
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled Cannabinoid receptor 1 using [3H]WIN-55212-2 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against G protein coupled human Cannabinoid receptor 2 using [3H]CP-55940 in HEK293 EBNA transfected cellsMore data for this Ligand-Target Pair