Affinity DataIC50: 7.80nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 920nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Daiichi Pharmaceutical
Curated by ChEMBL
Daiichi Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of Beta-adrenergic receptor kinase 1More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Daiichi Pharmaceutical
Curated by ChEMBL
Daiichi Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.57E+5nMAssay Description:Inhibition of Beta-adrenergic receptor kinase 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+5nMAssay Description:Concentration required to inhibit thrombin activity by 50%More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Daiichi Pharmaceutical
Curated by ChEMBL
Daiichi Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.63E+5nMAssay Description:Inhibition of Beta-adrenergic receptor kinase 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Concentration required to inhibit thrombin activity by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+6nMAssay Description:Concentration required to inhibit thrombin activity by 50%More data for this Ligand-Target Pair