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Found 137 with Last Name = 'gelhaus' and Initial = 'c'
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322349((R)-Methyl4-(2-(3-((adamantan-1-ylcarbamoyloxy)met...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322349((R)-Methyl4-(2-(3-((adamantan-1-ylcarbamoyloxy)met...)
Affinity DataKi:  14nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50257018((E)-methyl4-(2-((R,Z)-3-((4-chloro-2-(trifluoromet...)
Affinity DataKi:  17nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318713((2S,15S,18S,21S,24S)-15-(3-amino-3-oxopropyl)-2-be...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322342((R)-Methyl4-(2-(7-chloro-3-((4-chloro-2-(trifluoro...)
Affinity DataKi:  87nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314131((S,E)-Ethyl 4-((R)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  140nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314126((S)-Benzyl-2-[(Z)-3-((S)-1-benzyloxycarbonyl-2-phe...)
Affinity DataKi:  150nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  200nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataKi:  290nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assay in presence of de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318714((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314130((S)-2-[(E)-3-((S)-1-Benzyloxycarbonyl-2-phenylethy...)
Affinity DataKi:  340nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50325650(CHEMBL1224170 | S-isopentyl 3-methylbutane-1-sulfi...)
Affinity DataKi:  360nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318711((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assay in presence of d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322342((R)-Methyl4-(2-(7-chloro-3-((4-chloro-2-(trifluoro...)
Affinity DataKi:  460nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322343((R)-Methyl4-(2-(5-(4-bromophenyl)-3-((4-chloro-2-(...)
Affinity DataKi:  470nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  470nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50321811((4-Chloro-2-trifluoromethyl-phenyl)-carbamic acid ...)
Affinity DataKi:  700nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 to 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50321812((4-Chloro-2-trifluoromethyl-phenyl)-carbamic acid ...)
Affinity DataKi:  800nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 to 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50257018((E)-methyl4-(2-((R,Z)-3-((4-chloro-2-(trifluoromet...)
Affinity DataKi:  810nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304289(1-(4-Methoxyphenyl)-6,7-methylenedioxy-2-(4-methyl...)
Affinity DataKi:  850nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50257017((4-Chloro-2-trifluoromethyl-phenyl)-carbamic acid ...)
Affinity DataKi:  850nMAssay Description:Inhibition of cathepsin B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322341(CHEMBL1171803 | Methyl4-(2-((R)-3-((4-chloro-2-(tr...)
Affinity DataKi:  870nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322346((R)-Methyl4-(2-(3-((naphthalen-1-ylcarbamoyloxy)me...)
Affinity DataKi:  930nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318715((2S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,21-d...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50325651(CHEMBL1224171 | S-hexyl hexane-1-sulfinothioate)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318716((2S,8S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,2...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314128((S,E)-Methyl 2-(4-Ethoxy-4-oxobut-2-enamido)-5-oxo...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314127((S)-Benzyl-2-{(Z)-3-[(S)-1-((S)-1-benzyloxycarbony...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322343((R)-Methyl4-(2-(5-(4-bromophenyl)-3-((4-chloro-2-(...)
Affinity DataKi:  1.56E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318717((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257017((4-Chloro-2-trifluoromethyl-phenyl)-carbamic acid ...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of cathepsin L (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304288(2-(4-Acetylphenylureido)-1-(4-methoxyphenyl)-6,7-m...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322341(CHEMBL1171803 | Methyl4-(2-((R)-3-((4-chloro-2-(tr...)
Affinity DataKi:  2.22E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50322345((R)-Methyl4-(2-(3-((4-methoxyphenylcarbamoyloxy)me...)
Affinity DataKi:  2.23E+3nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50325648(CHEMBL1224167 | S-benzyl phenylmethanesulfinothioa...)
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50322347((R)-Methyl4-(2-(3-((butylcarbamoyloxy)methyl)-2-ox...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318709((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257015((4S)-4-{2-[3-(4-Chloro-2-trifluoromethyl-phenylcar...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of cathepsin L (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257019((4-Chloro-2-trifluoromethyl-phenyl)-carbamic acid ...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of cathepsin L (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50304290(2-Amino-6,7-dibenzyloxy-1-(4-methoxyphenyl)-2Hisoq...)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50325650(CHEMBL1224170 | S-isopentyl 3-methylbutane-1-sulfi...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50322346((R)-Methyl4-(2-(3-((naphthalen-1-ylcarbamoyloxy)me...)
Affinity DataKi:  3.48E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Universit£

Curated by ChEMBL
LigandPNGBDBM50314124((S,E)-ethyl 4-(tert-butoxycarbonylamino)-7-oxo-7-(...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assay in presence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50304288(2-(4-Acetylphenylureido)-1-(4-methoxyphenyl)-6,7-m...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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