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Found 468 with Last Name = 'geng' and Initial = 'b'
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284790(CHEMBL35987 | Sodium; (2S,5R)-3,3-dimethyl-7-oxo-6...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50033680(CHEMBL268919 | Sodium; (R)-3-acetoxymethyl-7-[1-te...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284783(CHEMBL37794 | Sodium; (R)-3-acetoxymethyl-7-methyl...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae SC 12368 E-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284783(CHEMBL37794 | Sodium; (R)-3-acetoxymethyl-7-methyl...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284786(CHEMBL36657 | Sodium; (R)-3-acetoxymethyl-7-[1-met...)
Affinity DataIC50:  37nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Celator Pharmaceuticals

US Patent
LigandPNGBDBM350085(3-[3-[4-[dideuterio(methylamino)methyl]phenyl]isox...)
Affinity DataIC50:  42nMAssay Description:Estimated IC50 values are as follows (obtained using STANDARD KINASEPROFILER).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284789((2S,5R,6Z)-6-(carboxymethylene)-3,3-dimethyl-7-oxo...)
Affinity DataIC50:  45nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284789((2S,5R,6Z)-6-(carboxymethylene)-3,3-dimethyl-7-oxo...)
Affinity DataIC50:  91nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae SC 12368 E-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284789((2S,5R,6Z)-6-(carboxymethylene)-3,3-dimethyl-7-oxo...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284794(CHEMBL36689 | Sodium; (R)-3-acetoxymethyl-5,5,8-tr...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284793(CHEMBL284539 | Sodium; (2S,5R)-6-[1-tert-butoxycar...)
Affinity DataIC50:  136nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284784(CHEMBL290112 | Sodium; (2S,5R)-6-[1-methoxycarbony...)
Affinity DataIC50:  154nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytes expressed as KonMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284794(CHEMBL36689 | Sodium; (R)-3-acetoxymethyl-5,5,8-tr...)
Affinity DataIC50:  260nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae SC 12368 E-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284784(CHEMBL290112 | Sodium; (2S,5R)-6-[1-methoxycarbony...)
Affinity DataIC50:  308nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
TBA

Curated by ChEMBL
LigandPNGBDBM50284790(CHEMBL35987 | Sodium; (2S,5R)-3,3-dimethyl-7-oxo-6...)
Affinity DataIC50:  361nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase TEM(Escherichia coli)
TBA

Curated by ChEMBL
LigandPNGBDBM50284792((6R,7Z)-3-[(acetyloxy)methyl]-7-(2-oxido-2-oxoethy...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate racemase(Helicobacter pylori J99)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50256537(1-(5-phenyl-3-(thiophen-2-yl)-3H-benzo[e][1,4]diaz...)
Affinity DataIC50:  500nMAssay Description:Inhibition of MurI in wild type Helicobacter pylori J99More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536589(US11242361, Compound 196)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536590(US11242361, Compound 197)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536591(US11242361, Compound 198)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536592(US11242361, Compound 199)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536593(US11242361, Compound 200)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536594(US11242361, Compound 201)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536595(US11242361, Compound 202)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536596(US11242361, Compound 203)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536597(US11242361, Compound 204)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536598(US11242361, Compound 205)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536599(US11242361, Compound 206)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536600(US11242361, Compound 207)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536601(US11242361, Compound 208)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536602(US11242361, Compound 209)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536603(US11242361, Compound 210)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536604(US11242361, Compound 296)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536605(4-(6-Bromo-2-methyl-3-(2-(piperidin-1-yl)acetyl)-1...)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536606(US11242361, Compound 298)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536607(US11242361, Compound 299)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536608(US11242361, Compound 300)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536609(US11242361, Compound 301)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536610(US11242361, Compound 302)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536611(US11242361, Compound 303)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536612(US11242361, Compound 304)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536613(US11242361, Compound 305)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536614(US11242361, Compound 306)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536615(US11242361, Compound 307)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536616(US11242361, Compound 308)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536617(US11242361, Compound 309)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536618(US11242361, Compound 310)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Proteostasis Therapeutics

US Patent
LigandPNGBDBM536619(US11242361, Compound 311 | US11242361, Compound 31...)
Affinity DataIC50:  550nMAssay Description:Using previously described methodology [B. H. Lee et al. Nature 2010, 467 (9), 179, the contents of which are expressly incorporated by reference her...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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