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Found 283 with Last Name = 'kim' and Initial = 'bm'
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  1nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50131716(CHEMBL430892 | [3-(4-Bromo-2-chloro-phenyl)-2,5-di...)
Affinity DataKi:  1.90nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  30nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  85nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  90nMAssay Description:Mixed type inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355372(CHEMBL482212)
Affinity DataKi:  250nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355361(CHEMBL1835541)
Affinity DataKi:  1.40E+3nMAssay Description:Non-Competitive inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Reversible inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  8.50E+4nMAssay Description:Reversible inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285450(CHEMBL300140 | [(1S,2R)-1-Benzyl-3-((S)-4-[2,2']bi...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285455(CHEMBL293992 | [(1S,2R)-3-((S)-4-Benzo[b]thiophen-...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285454(CHEMBL294392 | [(1S,2R)-1-Benzyl-3-((S)-2-tert-but...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285453(CHEMBL292193 | {(1S,2R)-1-Benzyl-3-[(S)-4-(4-bromo...)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285456(CHEMBL410311 | {(1S,2R)-1-Benzyl-3-[(S)-4-(5-bromo...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285459(CHEMBL301269 | [(1S,2R)-1-Benzyl-3-((S)-2-tert-but...)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285452(CHEMBL60697 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-buty...)
Affinity DataIC50:  0.470nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50283282(CHEMBL55586 | L-738872 | {(1S,2R)-1-Benzyl-3-[(S)-...)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285451(CHEMBL301260 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285458(CHEMBL57566 | [(1S,2R)-1-Benzyl-3-((S)-2-tert-buty...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285460(((1S,2R)-1-Benzyl-3-{(S)-2-tert-butylcarbamoyl-4-[...)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285277(CHEMBL72497 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-buty...)
Affinity DataIC50:  0.950nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285275(CHEMBL72399 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-buty...)
Affinity DataIC50:  1.10nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285274(CHEMBL307966 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50283288(CHEMBL72487 | [(1S,2R)-1-Benzyl-3-((S)-2-tert-buty...)
Affinity DataIC50:  1.30nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285276(CHEMBL307091 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285270(CHEMBL308410 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285449(CHEMBL57238 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-buty...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285271(CHEMBL72385 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-buty...)
Affinity DataIC50:  1.80nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50460108(CHEMBL4225016)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant human JAK1 (866-end residues) in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50283284(CHEMBL75310 | {(1S,2R)-1-Benzyl-3-[2-((R)-tert-but...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human JAK1 (866-end residues) in presence of ATPMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285272(CHEMBL306772 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  2.30nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285273(CHEMBL419072 | {(1S,2R)-1-Benzyl-3-[(S)-2-tert-but...)
Affinity DataIC50:  2.5nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 protease enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of recombinant GST-tagged human JAK1 (852 to 1142 residues) using IRS-1 as substrate in presence of 40 uM ATP by mobility shift assayMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50285457(CHEMBL56247 | [(1S,2R)-1-Benzyl-3-((S)-2-tert-buty...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50460106(CHEMBL4227132)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of recombinant human JAK1 (866-end residues) in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories

LigandPNGBDBM305((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  3.80nMAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM305((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  3.80nMAssay Description:Tested in vitro for the ability to inhibit HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50460114(CHEMBL4226840)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of recombinant human JAK1 (866-end residues) in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of recombinant GST-tagged human JAK2 (809 to 1153 residues) catalytic cytoplasmic domain expressed in baculovirus expression system using ...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories

LigandPNGBDBM300((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  4.80nMAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM300((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  4.80nMAssay Description:Tested in vitro for the ability to inhibit HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334431(CHEMBL1643873 | N-((3S,5R)-5-((N-hydroxyformamido)...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories

LigandPNGBDBM304((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  5.30nMAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM304((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  5.30nMAssay Description:Tested in vitro for the ability to inhibit HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeptide deformylase(Pseudomonas aeruginosa)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50334430(CHEMBL1643872 | N-((3S,5R)-5-((N-hydroxyformamido)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Pseudomonas aeruginosa peptide deformylase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM303((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  8.30nMAssay Description:Tested in vitro for the ability to inhibit HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Merck Research Laboratories

LigandPNGBDBM303((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  8.30nMAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM291((2R,3R)-1,1-dioxo-2-(propan-2-yl)--thiolan-3-yl N-...)
Affinity DataIC50:  8.40nMAssay Description:Tested in vitro for the ability to inhibit HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
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