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Found 397 with Last Name = 'koch' and Initial = 'o'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579476(US11485700, Compound (+)-CBD-HPE)
Affinity DataKi:  0.800nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579476(US11485700, Compound (+)-CBD-HPE)
Affinity DataKi:  3.10nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579474(US11485700, Compound (+)-CBD-GE)
Affinity DataKi:  12.9nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579473(US11485700, Compound (+)-CBD)
Affinity DataKi:  28nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579472(US11485700, Compound (+)-CBDV)
Affinity DataKi:  33.1nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM576352(US11485700, Compound (+)-CBD-ME)
Affinity DataKi:  40.5nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579472(US11485700, Compound (+)-CBDV)
Affinity DataKi:  294nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579473(US11485700, Compound (+)-CBD)
Affinity DataKi:  345nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM579474(US11485700, Compound (+)-CBD-GE)
Affinity DataKi:  359nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Symrise

US Patent
LigandPNGBDBM576352(US11485700, Compound (+)-CBD-ME)
Affinity DataKi:  982nMAssay Description:Membranes from human CB1 or CB2 receptor-transfected cells (RBHCB1M400UA and RBXCB2M400UA, respectively) were supplied by Perkin-Elmer Life and Analy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of neuraminidase H274Y mutant in Oseltamivir-resistant Influenza A virus A/Berlin/55/08(H1N1) using Na-star as substrate preincubated for ...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.660nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.75nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50028503(CHEMBL81717 | Guanidino-Oseltamivir Carboxylicacid)
Affinity DataIC50:  0.990nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataIC50:  1.10nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242179(CHEMBL4093459)
Affinity DataIC50:  1.60nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)
Affinity DataIC50:  1.70nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242168(CHEMBL4101206)
Affinity DataIC50:  1.90nMAssay Description:Concentration required to inhibit the activity of gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
European Institute For Molecular Imaging (Eimi)

Curated by ChEMBL
LigandPNGBDBM50585247(CHEMBL5079389)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced inward current at -60 mV preincubated for 30 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
European Institute For Molecular Imaging (Eimi)

Curated by ChEMBL
LigandPNGBDBM50585247(CHEMBL5079389)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced inward current at -60 mV preincubated for 30 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242190(CHEMBL4103644)
Affinity DataIC50:  2nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50345596(4-methyl-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(...)
Affinity DataIC50:  2.10nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242167(CHEMBL4076193)
Affinity DataIC50:  2.10nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50496023(CHEMBL3120197)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242161(CHEMBL4097771)
Affinity DataIC50:  2.30nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50242166(CHEMBL4085713)
Affinity DataIC50:  2.5nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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