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Found 44 with Last Name = 'kouji' and Initial = 'h'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151161(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  220nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataKi:  244nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151159(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  280nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186371(CHEMBL264120 | c(his-D-phe-arg-trp-Aoc))
Affinity DataKi:  319nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186370(CHEMBL379627 | c(his-D-phe-arg-trp-Ahx))
Affinity DataKi:  670nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151163(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  870nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151168(5-Phenyl-1H-pyrrole-2-carboxylic acid (cyclohexylc...)
Affinity DataKi:  910nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151160(5-Phenyl-1H-pyrrole-2-carboxylic acid (3-diethylam...)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151169(5-Phenyl-1H-pyrrole-2-carboxylic acid [1-cyclohexy...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151158(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-tert-buty...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151167(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.29E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151164(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.32E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151157(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  1.37E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151165(5-Phenyl-1H-pyrrole-2-carboxylic acid (1-cyclohexy...)
Affinity DataKi:  1.92E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151170(CHEMBL185887 | N-[Cyclohexylcarbamoyl-(4-fluoro-ph...)
Affinity DataKi:  2.03E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151166(5-Phenyl-1H-pyrrole-2-carboxylic acid [cyclohexylc...)
Affinity DataKi:  2.63E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186366(CHEMBL211131 | c(his-L-phe-arg-trp-Aoc))
Affinity DataKi:  4.42E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186368(CHEMBL379531 | c(his-D-phe-arg-trp-Abu))
Affinity DataKi:  5.78E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research

Curated by ChEMBL
LigandPNGBDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304254((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304255((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  13.2nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304256((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  10.1nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304257((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  75.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304258((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  20.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304253((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  8.51nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304252((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  6.94nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186371(CHEMBL264120 | c(his-D-phe-arg-trp-Aoc))
Affinity DataEC50:  77.4nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataEC50:  67nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186370(CHEMBL379627 | c(his-D-phe-arg-trp-Ahx))
Affinity DataEC50:  3.12E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  72.9nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186370(CHEMBL379627 | c(his-D-phe-arg-trp-Ahx))
Affinity DataEC50:  1.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186368(CHEMBL379531 | c(his-D-phe-arg-trp-Abu))
Affinity DataEC50:  1.58E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186372(CHEMBL380198 | c(his-D-phe-arg-trp-betaala))
Affinity DataEC50:  1.11E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Affinity DataEC50:  15.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186372(CHEMBL380198 | c(his-D-phe-arg-trp-betaala))
Affinity DataEC50:  135nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186369(CHEMBL210399 | c(his-D-phe-arg-trp-Ava))
Affinity DataEC50:  3.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304259((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  16.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  1.80nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186369(CHEMBL210399 | c(his-D-phe-arg-trp-Ava))
Affinity DataEC50:  1.01E+4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186368(CHEMBL379531 | c(his-D-phe-arg-trp-Abu))
Affinity DataEC50:  270nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186366(CHEMBL211131 | c(his-L-phe-arg-trp-Aoc))
Affinity DataEC50:  9.59E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186366(CHEMBL211131 | c(his-L-phe-arg-trp-Aoc))
Affinity DataEC50:  5.10E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186371(CHEMBL264120 | c(his-D-phe-arg-trp-Aoc))
Affinity DataEC50:  16.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed