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Found 35 with Last Name = 'laube' and Initial = 'm'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50272095(4-(3-(4-methoxyphenyl)-1H-indol-2-yl)benzenesulfon...)
Affinity DataIC50:  6nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50272096(3-(4-methoxyphenyl)-2-(4-(methylsulfonyl)phenyl)-1...)
Affinity DataIC50:  20nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50272131(3-(4-fluorophenyl)-2-(4-(methylsulfonyl)phenyl)-1H...)
Affinity DataIC50:  20nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant COX2 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50272131(3-(4-fluorophenyl)-2-(4-(methylsulfonyl)phenyl)-1H...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant COX2 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50272131(3-(4-fluorophenyl)-2-(4-(methylsulfonyl)phenyl)-1H...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of ovine COX1 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of ovine COX1 by enzymatic fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584200(CHEMBL5083438)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584201(CHEMBL5091965)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584202(CHEMBL5085479)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584204(CHEMBL5082631)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584205(CHEMBL5072994)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584206(CHEMBL5088591)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584207(CHEMBL5091083)
Affinity DataKd:  340nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584208(CHEMBL5071902)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584209(CHEMBL5094773)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584210(CHEMBL5079936)
Affinity DataKd:  7.00E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584211(CHEMBL5093259)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584212(CHEMBL5074099)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584213(CHEMBL5078753)
Affinity DataKd:  8.00E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584214(CHEMBL5082399)
Affinity DataKd:  230nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant using N-alpha-(6-FAM)-N-epsilon-(4-Iodophenylbutanoyl)-D-lysine as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584198(CHEMBL5078842)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584194(CHEMBL5089368)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584199(CHEMBL5093073)
Affinity DataKd:  360nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584198(CHEMBL5078842)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584197(CHEMBL5093280)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584196(CHEMBL5075340)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584195(CHEMBL5093981)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584194(CHEMBL5089368)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Institute Of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584203(CHEMBL5091156)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed