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Found 113 with Last Name = 'le' and Initial = 'tv'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289438((4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-1-(3-hydr...)
Affinity DataKi:  0.0580nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289443((4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-1-(3-hydr...)
Affinity DataKi:  0.0810nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289441((4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-1-(4-hydr...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289445((4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-1-(5-hydr...)
Affinity DataKi:  0.240nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKi:  0.240nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM150((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis({...)
Affinity DataKi:  0.340nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM33((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(6...)
Affinity DataKi:  0.470nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289440((4R,5S,6S,7R)-1,4,7-Tribenzyl-5,6-dihydroxy-3-(5-h...)
Affinity DataKi:  0.680nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289437(3-[(4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-3-(5-h...)
Affinity DataKi:  0.720nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM25((4R,5S,6S,7R)-4,7-dibenzyl-1-(cyclopropylmethyl)-5...)
Affinity DataKi:  0.990nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM28((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(5...)
Affinity DataKi:  1.40nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289439((4R,5S,6S,7R)-4,7-Dibenzyl-5,6-dihydroxy-1-(6-hydr...)
Affinity DataKi:  1.70nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50289446(CHEMBL280989 | N-(5-{(4R,5S,6S,7R)-4,7-Dibenzyl-5,...)
Affinity DataKi:  8.90nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM67(DMPC Cyclic Urea 47 | N-{5-[(4R,5S,6S,7R)-4,7-dibe...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM69(CHEMBL282395 | DMPC Cyclic Urea 49 | N-{5-[(4R,5S,...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM70(DMPC Cyclic Urea 50 | N-{5-[(4R,5S,6S,7R)-4,7-dibe...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM76(DMPC Cyclic Urea 56 | methyl 6-[(4R,5S,6S,7R)-4,7-...)
Affinity DataKi:  29nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM81((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(7...)
Affinity DataKi:  34nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM87((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(4...)
Affinity DataKi:  42nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM92((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(3...)
Affinity DataKi:  51nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM93(DMPC Cyclic Urea 73 | N-{5-[(4R,5S,6S,7R)-4,7-dibe...)
Affinity DataKi:  59nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM98((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(5...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM114(1-{5-[(4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-3-{...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM108(DMPC Cyclic Urea 88 | N-{5-[(4R,5S,6S,7R)-4,7-dibe...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM117(DMPC Cyclic Urea 97 | N-{5-[(4R,5S,6S,7R)-4,7-dibe...)
Affinity DataKi:  350nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM120((4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis(8...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM128((4R,5S,6S,7R)-1,3-bis(4-aminobutyl)-4,7-dibenzyl-5...)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM127((4R,5S,6S,7R)-1,3-bis(5-aminopentyl)-4,7-dibenzyl-...)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50433097(CHEMBL2377258)
Affinity DataIC50:  77nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50220856(2-(3-(4-phenylpiperidin-1-yl)propyl)quinazolin-4(3...)
Affinity DataIC50:  79nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50433098(CHEMBL2377257)
Affinity DataIC50:  189nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50220864(2-(3-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-...)
Affinity DataIC50:  304nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50433095(CHEMBL2377260)
Affinity DataIC50:  388nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50433096(CHEMBL2377259)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311577(CHEMBL561967 | Erybreadin B | erybraedin B)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50104694((R)-4-hydroxy-5-(hydroxymethyl)-3-palmitoylfuran-2...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311580(CHEMBL1087148 | Erybreadin D)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311582(CHEMBL1086765 | Erybreadin C)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50317432(CHEMBL1098728 | NEORAUTENOL)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311579(CHEMBL551155 | folitenol)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311581(CHEMBL1086764 | erysubin E)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Sungkyunkwan [Corrected] University

Curated by ChEMBL
LigandPNGBDBM50433099(CHEMBL2377256)
Affinity DataIC50:  8.89E+3nMAssay Description:Inhibition of PARP1 (unknown origin) after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311572(CHEMBL1076430 | Erythribyssin A)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311578(3,9-Dihydroxy-4-prenyl-[6aR;11aR]pterocarpan | CHE...)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311586(CHEMBL1088462 | erystagallin A)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311583(Abyssinone II | CHEMBL508534 | phaseolidin | phase...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311575(CHEMBL1079408 | Eryvarin K)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311574(CHEMBL1079407 | Erythribyssin C)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chosun University

Curated by ChEMBL
LigandPNGBDBM50311573(CHEMBL1079406 | Erythribyssin B)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant PTP1B assessed as p-nitrophenol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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