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Found 83 with Last Name = 'leiros' and Initial = 'hk'
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129065(CHEMBL3278535)
Affinity DataKi:  1.86E+5nMAssay Description:Competitive inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129065(CHEMBL3278535)
Affinity DataKi:  1.86E+5nMAssay Description:Competitive inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50174202(2-benzoylbenzoic acid | CHEMBL196812)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129030(CHEMBL81936)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129032(CHEMBL82115)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195796(CHEMBL3910343)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataIC50:  4.98E+4nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195795(CHEMBL3908259)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM114408(2-(7-chloranylquinolin-4-yl)sulfanylethanoic acid ...)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM114408(2-(7-chloranylquinolin-4-yl)sulfanylethanoic acid ...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129035(CHEMBL1778133)
Affinity DataIC50:  2.32E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195792(CHEMBL3896367)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195789(CHEMBL3967375)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195794(CHEMBL3913021)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195793(CHEMBL123234)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM73278(4-keto-4-(4-propylphenyl)butyric acid | 4-oxidanyl...)
Affinity DataIC50:  2.87E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129082(CHEMBL1324612)
Affinity DataIC50:  2.98E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129066(CHEMBL3627736)
Affinity DataIC50:  3.14E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129065(CHEMBL3278535)
Affinity DataIC50:  4.79E+5nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129081(CHEBI:33070 | Indole-3-Butyric Acid)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129065(CHEMBL3278535)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50355012(CHEMBL1834963)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50442179(CHEMBL2441619)
Affinity DataIC50:  5.92E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129081(CHEBI:33070 | Indole-3-Butyric Acid)
Affinity DataIC50:  7.57E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50060966(4-Phenoxy-benzoic acid | CHEMBL107518 | US10322118...)
Affinity DataIC50:  8.70E+5nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129079(CHEMBL3629240)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129031(CHEMBL1879588)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195790(CHEMBL3951674)
Affinity DataIC50:  1.02E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM114408(2-(7-chloranylquinolin-4-yl)sulfanylethanoic acid ...)
Affinity DataIC50:  1.23E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM114408(2-(7-chloranylquinolin-4-yl)sulfanylethanoic acid ...)
Affinity DataIC50:  1.24E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195791(CHEMBL2018158)
Affinity DataIC50:  1.39E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129065(CHEMBL3278535)
Affinity DataIC50:  1.43E+6nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129081(CHEBI:33070 | Indole-3-Butyric Acid)
Affinity DataIC50:  1.95E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129081(CHEBI:33070 | Indole-3-Butyric Acid)
Affinity DataIC50:  1.95E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50121955(4-Phenyl-pyridine | CHEMBL109074 | US11634391, Com...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM197302(Benzoic acid | SAMPL4, O1)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195798(CHEMBL3931620)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50195797(CHEMBL3950623)
Affinity DataIC50:  2.20E+6nMAssay Description:Inhibition of native signal containing Klebsiella pneumoniae OXA-48 using nitrocefin substrate pre-incubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129069(CHEMBL3629239)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition of Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) using nitrocefin as substrate prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM73278(4-keto-4-(4-propylphenyl)butyric acid | 4-oxidanyl...)
Affinity DataIC50:  3.09E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Klebsiella pneumoniae)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM73278(4-keto-4-(4-propylphenyl)butyric acid | 4-oxidanyl...)
Affinity DataIC50:  3.11E+6nMAssay Description:Inhibition of His-tagged Klebsiella pneumoniae NDM-1 expressed in Escherichia coli BL21-AI cells using imipinem as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129062(CHEBI:43968 | ICI-194660 | Meropenem | Merrem | Me...)
Affinity DataKd:  1.20E+4nMAssay Description:Reversible binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataKon:  0.0250M-1s-1Assay Description:Reversible binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 s...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129035(CHEMBL1778133)
Affinity DataKd:  1.45E+5nMAssay Description:Binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 secs by SPR ...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50129032(CHEMBL82115)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 secs by SPR ...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM73278(4-keto-4-(4-propylphenyl)butyric acid | 4-oxidanyl...)
Affinity DataKd:  1.73E+5nMAssay Description:Binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 secs by SPR ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM114408(2-(7-chloranylquinolin-4-yl)sulfanylethanoic acid ...)
Affinity DataKd:  2.64E+5nMAssay Description:Binding affinity to Pseudomonas aeruginosa 301-5473 metallo-beta-lactamase VIM-2 expressed in Escherichia coli BL21(DE3) measured for 15 secs by SPR ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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