TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 4.05E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 5.41E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 6.38E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human URAT1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine
Curated by ChEMBL
Hunan University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 7.84E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University
Curated by ChEMBL
Tianjin Medical University
Curated by ChEMBL
Affinity DataIC50: 3.65E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 3.93E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 4.18E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.25E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.43E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.59E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.68E+5nMAssay Description:Reactivation of sarin-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 6.26E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 6.37E+5nMAssay Description:Reactivation of VX-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 mins f...More data for this Ligand-Target Pair
Affinity DataIC50: 6.58E+5nMAssay Description:Reactivation of tabun-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 min...More data for this Ligand-Target Pair
Affinity DataIC50: 6.68E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 6.85E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair