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Found 40 with Last Name = 'maccari' and Initial = 'g'
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254171(CHEMBL4069120)
Affinity DataKi:  220nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352509(CHEMBL1824848)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352515(CHEMBL1824850)
Affinity DataKi:  9.30E+3nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM60660(2-[8-(6-amino-1H-benzimidazol-2-yl)octyl]-3H-benzi...)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352513(CHEMBL1824853)
Affinity DataKi:  1.11E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352512(CHEMBL1824852)
Affinity DataKi:  1.18E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352510(CHEMBL1824849)
Affinity DataKi:  1.31E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352508(CHEMBL1824847)
Affinity DataKi:  1.31E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254176(CHEMBL3040884)
Affinity DataKi:  1.41E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254177(CHEMBL3040820)
Affinity DataKi:  1.78E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352514(CHEMBL1824854)
Affinity DataKi:  2.23E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Universit£

Curated by ChEMBL
LigandPNGBDBM50352511(CHEMBL1824851)
Affinity DataKi:  2.69E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR using trypanothione as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254178(CHEMBL3558827)
Affinity DataKi:  3.13E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254180(CHEMBL3558806)
Affinity DataKi:  3.48E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254181(CHEMBL3558803)
Affinity DataKi:  3.58E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254182(CHEMBL3040830)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254179(CHEMBL3558802)
Affinity DataKi:  4.53E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254183(CHEMBL575667)
Affinity DataKi:  5.08E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  600nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  670nMAssay Description:Inhibition of human MDR1 expressed in mouse L5178 cells assessed as increase in intracellular accumulation of rhodamine 123 by FACSCalibur flow cytom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254171(CHEMBL4069120)
Affinity DataIC50:  680nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484507(CHEMBL1927604)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378908(CHEMBL1688197)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human MDR1 expressed in mouse L5178 cells assessed as increase in intracellular accumulation of rhodamine 123 by FACSCalibur flow cytom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484506(CHEMBL1927602)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484511(CHEMBL1927605)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484510(CHEMBL1927606)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484509(CHEMBL1927603)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484505(CHEMBL1927601)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50484508(CHEMBL1927607)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50339000((1R,2R,9R)-2-methoxy-9-((2-methoxyethoxy)methoxy)-...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human MDR1 expressed in mouse L5178 cells assessed as increase in intracellular accumulation of rhodamine 123 by FACSCalibur flow cytom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254176(CHEMBL3040884)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254177(CHEMBL3040820)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254178(CHEMBL3558827)
Affinity DataIC50:  9.70E+4nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254180(CHEMBL3558806)
Affinity DataIC50:  1.08E+5nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254181(CHEMBL3558803)
Affinity DataIC50:  1.11E+5nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254182(CHEMBL3040830)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254179(CHEMBL3558802)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChitinase(Hypocrea rufa)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50254183(CHEMBL575667)
Affinity DataIC50:  1.57E+5nMAssay Description:Inhibition of Trichoderma viride chitinase incubated for 10 mins to 3 hrs using 4-nitrophenyl N-acetyl-beta-D-glucosaminide substrate by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50036568(CHEMBL3353611)
Affinity DataKd:  2.65E+4nMAssay Description:Binding affinity to human serum albumin after 30 mins by fluorescence spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed