Affinity DataKi: 0.0300nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.580nMAssay Description:Binding affinity to sigma 2 receptor in human MCF7 cells assessed as displacement of compound by measuring inhibition constant of DTG incubated for 1...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.680nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes assessed as inhibition constant by Wallac 1450 MicroBeta liqu...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.90nMAssay Description:Binding affinity to human CB2 receptor stably expressed in HEK cells assessed as inhibition constant by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity to sigma 2 receptor in human MCF7 cells assessed as displacement of compound by measuring inhibition constant of DTG incubated for 1...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by liquid sc...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.10nMAssay Description:Binding affinity to sigma 2 receptor in human MCF7 cells assessed as displacement of compound by measuring inhibition constant of 2-(3-(6,7-dimethoxy...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.5nMAssay Description:Binding affinity to human CB2 receptor stably expressing HEK cells assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to sigma 2 receptor in human MCF7 cells assessed as displacement of compound by measuring inhibition constant of 2-(3-(6,7-dimethoxy...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.40nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 6.90nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in HEK cell membrane measured after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 10nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 11nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]RHM-1 from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 12nMAssay Description:Binding affinity to human recombinant CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to CB2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 14nMAssay Description:Displacement of [3H]RHM-1 from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 14nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by liquid sc...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 18nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]HU-243 binding to CB2 receptor in human COS-7 cellsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 27nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 30nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 37nMAssay Description:Binding affinity to human CB2 receptor stably expressed in HEK cells assessed as inhibition constant by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 39nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 39nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 40nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 51nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 51nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 62nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 89nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 93nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 93.4nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Binding affinity to human CB2 receptor stably expressed in HEK cells assessed as inhibition constant by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info