BindingDB PrimarySearch

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50217952((1R,5R,9S)-(-)-9-hydroxy-5-(3-hydroxyphenyl-2-phen...)

Ki: 0.190nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50217956((1R,5S)-(+)-5-(3-hydroxyphenyl)-9-methylene-2-phen...)

Ki: 0.190nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530711(CHEMBL4553052)

Ki: 0.191nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530711(CHEMBL4553052)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50001019(6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,...)

Ki: 0.200nMAssay Description:Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530731(CHEMBL4580446)

Ki: 0.240nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530731(CHEMBL4580446)

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50041240((6S,11R)-3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahyd...)

Ki: 0.300nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095694(3-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2...)

Ki: 0.400nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095706(4-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2...)

Ki: 0.400nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50037492(CHEMBL113995 | [(S)-2-(2-{(S)-2-[(S)-2-Amino-3-(4-...)

Ki: 0.460nMAssay Description:Binding affinity against opioid receptor by displacing radioligand [3H]DAMGOMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095705(3-But-2-ynyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 0.5nMAssay Description:Ki value determined against Opioid receptor mu 1 using [3H]-DAMGO at the Kd concentration 0.57 nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530712(CHEMBL4591248)

Ki: 0.501nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530712(CHEMBL4591248)

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530712(CHEMBL4591248)

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530712(CHEMBL4591248)

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50217950((1R,5S,9R)-(+)-5-(3-hydroxyphenyl)-9-methyl-2-phen...)

Ki: 0.600nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Kappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50217956((1R,5S)-(+)-5-(3-hydroxyphenyl)-9-methylene-2-phen...)

Ki: 0.650nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50041240((6S,11R)-3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahyd...)

Ki: 0.900nMAssay Description:Ki value determined against Opioid receptor mu 1 using [3H]-DAMGO at the Kd concentration 0.57 nMMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

Sigma non-opioid intracellular receptor 1(RAT)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095699(3-Hex-5-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 1.10nMAssay Description:Ki value determined against Sigma opioid receptor type 1 using [(+)-[3H]pentazocaine at the Kd concentration 2nM .More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50381677(CHEMBL1256748 | U-69593)

Ki: 1.20nMAssay Description:Binding affinity against opioid receptor by displacing radioligand [3HlU69,593More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 1.30nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095707(3-But-3-ynyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 1.40nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50001036(3-(3-Chloro-allyl)-6,11-dimethyl-1,2,3,4,5,6-hexah...)

Ki: 1.5nMAssay Description:Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50037478((6S,11R)-6,11-Dimethyl-3-propyl-1,2,3,4,5,6-hexahy...)

Ki: 1.5nMAssay Description:Inhibition against mu receptor from displacement studies using 0.5 nM [3H]-DAMGO in rhesus monkey cortex membraneMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530723(CHEMBL4455627)

Ki: 1.90nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530723(CHEMBL4455627)

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50037489((6S,11S)-3-Heptyl-6,11-dimethyl-1,2,3,4,5,6-hexahy...)

Ki: 1.90nMAssay Description:Inhibition against sigma receptor using displacement of 3 nM [3H]pentazocine in homogenate of guinea pig brain cerebellumMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50367061(NALORPHINE | NALORPHINE HYDROCHLORIDE)

Ki: 2nMAssay Description:Compound administered subcutaneously was evaluated for inhibition constant measured as the displacement of [3H]DAGO from rat brainMore data for this Ligand-Target Pair

Purchase KEGG PC cid PC sid Similars

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Kappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50037478((6S,11R)-6,11-Dimethyl-3-propyl-1,2,3,4,5,6-hexahy...)

Ki: 2nMAssay Description:Inhibition against kappa receptor from displacement studies using 1.5 nM [3H]U-69593 in rhesus monkey cortex membraneMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

Sigma non-opioid intracellular receptor 1(RAT)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095711(6,11-Dimethyl-3-pent-4-enyl-1,2,3,4,5,6-hexahydro-...)

Ki: 2.10nMAssay Description:Ki value determined against Sigma opioid receptor type 1 using [(+)-[3H]pentazocaine at the Kd concentration 2nM .More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095703(3-But-3-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 2.10nMAssay Description:Ki value determined against Opioid receptor mu 1 using [3H]-DAMGO at the Kd concentration 0.57 nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50037476((6R,11S)-3-Hexyl-6,11-dimethyl-1,2,3,4,5,6-hexahyd...)

Ki: 2.30nMAssay Description:Inhibition against sigma receptor using displacement of 3 nM [3H]pentazocine in homogenate of guinea pig brain cerebellumMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530737(CHEMBL4449355)

Ki: 2.60nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530737(CHEMBL4449355)

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50037484((6S,11S)-6,11-Dimethyl-3-octyl-1,2,3,4,5,6-hexahyd...)

Ki: 2.80nMAssay Description:Inhibition against sigma receptor using displacement of 3 nM [3H]pentazocine in homogenate of guinea pig brain cerebellumMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)

Ki: 3nMAssay Description:Binding affinity against opioid receptor by displacing radioligand [3H]DPDPEMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50001039(6,11-Dimethyl-3-(1-methyl-allyl)-1,2,3,4,5,6-hexah...)

Ki: 3nMAssay Description:Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50067447(3-((R)-9-Methyl-2-phenethyl-2-aza-bicyclo[3.3.1]no...)

Ki: 3.10nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

CHEMBL PC cid PC sid Patents Similars

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50037482((6S,11R)-3-Butyl-6,11-dimethyl-1,2,3,4,5,6-hexahyd...)

Ki: 3.40nMAssay Description:Inhibition against mu receptor from displacement studies using 0.5 nM [3H]-DAMGO in rhesus monkey cortex membraneMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530724(CHEMBL4519184)

Ki: 3.40nMAssay Description:Inhibition of N-terminal His6-tagged wild type human NNMT expressed in Escherichia coli NiCo21(DE3) assessed as reduction in 1-methylquinolinium leve...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Nicotinamide N-methyltransferase(Homo sapiens (Human))
Biokin

Curated by ChEMBL

BDBM50530724(CHEMBL4519184)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50001031(3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-me...)

Ki: 3.60nMAssay Description:Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50037480((6R,11S)-6,11-Dimethyl-3-pentyl-1,2,3,4,5,6-hexahy...)

Ki: 3.80nMAssay Description:Inhibition against sigma receptor using displacement of 3 nM [3H]pentazocine in homogenate of guinea pig brain cerebellumMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Kappa-type opioid receptor(Mus musculus (Mouse))
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095705(3-But-2-ynyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)

Ki: 3.90nMAssay Description:Ki value determined against Opioid receptor kappa 1 using [3H]U69, 593 at the Kd concentration 0.95 nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Kappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50217950((1R,5S,9R)-(+)-5-(3-hydroxyphenyl)-9-methyl-2-phen...)

Ki: 4nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL

BDBM50001046(6,11-Dimethyl-3-(4-phenyl-butyl)-1,2,3,4,5,6-hexah...)

Ki: 4nMAssay Description:Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Mu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL

BDBM50095694(3-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2...)

Ki: 4.20nMAssay Description:Ki value determined against Opioid receptor mu 1 using [3H]-DAMGO at the Kd concentration 0.57 nMMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Mu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL

BDBM50037469((6S,11R)-3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,...)

Ki: 4.20nMAssay Description:Inhibition against mu receptor from displacement studies using 0.5 nM [3H]-DAMGO in rhesus monkey cortex membraneMore data for this Ligand-Target Pair