Compile Data Set for Download or QSAR
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Found 262 with Last Name = 'mays' and Initial = 'r'
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197025(CHEMBL439904 | PYY(3-36))
Affinity DataKi:  0.400nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208974(CHEMBL390543 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208948(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198507(2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198532(1-(2-chlorophenyl)-2-(4-chlorophenyl)-5-cyclohexyl...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197011(CHEMBL238533 | PYY(22-36))
Affinity DataKi:  3nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198519(1-(2-chlorophenyl)-2-(4-chlorophenyl)-3-methyl-5-(...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208975(1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50140237(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imi...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197010((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  4nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197019((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  4nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197010((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]PYY from human NPY2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198526(5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208955(2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imida...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208951(CHEMBL229583 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50205093(CHEMBL428017 | LRHYLNLLTRQRY-NH2)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]PYY from human NPY2 receptor in KAN-TS cells by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197023((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  5nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208968(2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198529(5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(3,4-dimetho...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208972(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197009((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  6nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197021((2S)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoy...)
Affinity DataKi:  6nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197020((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  6nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197022((2S)-2-[(2S)-2-[(2S,3R)-2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  6nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198525(5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-fluorophe...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208969(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208978(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208973(1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphe...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198513(2-(4-chlorophenyl)-5-cyclohexyl-1-(2,4-dichlorophe...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198516(1-(2-chlorophenyl)-5-cyclohexyl-2-(4-methoxyphenyl...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50123692(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyr...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198511(5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-methoxyph...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50319488(CHEMBL1084901 | rac-{5-Chloro-3-[2-(3,5-dimethyl-i...)
Affinity DataKi:  8nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50205095((S)-2-((S)-2-((2S,3R)-2-((S)-2-((S)-2-((S)-2-((S)-...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [125I]PYY from human NPY2 receptor in KAN-TS cells by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208956(CHEMBL229584 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208982(2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50091668(AcPYY(22-36) | CHEMBL269267 | N-alpha-Ac-PYY(22-36...)
Affinity DataKi:  9nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198535(5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50198517(5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-p-t...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208971(5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50210327((2S)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoy...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]PYY from human NPY2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50319486(CHEMBL1084893 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50319487(CHEMBL1084894 | rac-{2-Methyl-3-[2-(3-methyl-5-phe...)
Affinity DataKi:  13nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50162903(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208976(CHEMBL395322 | rac-2-(2-chlorophenyl)-1-(4-chlorop...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208970(2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohe...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50319482(CHEMBL1082939 | rac-{3-[2-(3,5-Dimethyl-isoxazol-4...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human prostaglandin D2 receptor by cell based radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208979(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197017((2S)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoy...)
Affinity DataKi:  18nMAssay Description:Displacement of human [125I]PYY from NPY2 receptor expressed in human KAN-TS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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