Affinity DataKi: 300nMAssay Description:Binding affinity against angiotensin II receptor type 2 (AT2) of rat adrenal medulla.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0320nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]-ET-1 binding to rat aorta membrane Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibition of [125I]-ET-1 binding to rat aorta membrane Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against AT1 receptor of rat adrenal cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against AT1 receptor of rat adrenal cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Ability to displace [125I]-Endothelin-1 from endothelin B receptor in porcine kidney membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:In vitro ability to inhibit specific [125I]ET1 binding to rat aorta membranes Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:In vitro binding affinity determined against angiotensin II AT1 receptor in rat adrenal cortex preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair