TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 16.3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 256nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 449nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 449nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 487nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.79E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 6.76E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 8.73E+3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 8.73E+3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 4.64E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 4.64E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against human Cholecystokinin type B receptor in CHO-K1 cells using [125I]-Bolton-Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 0.890nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Glaxo Wellcome Research And Development
Curated by ChEMBL
Glaxo Wellcome Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against human Cholecystokinin type A receptor in membrane preparation isolated from CHO-K1 cells stably transfected with cDNA of hum...More data for this Ligand-Target Pair
Affinity DataIC50: <2nMpH: 9.5 T: 2°CAssay Description:Selection of DNA-encoded libraries (DELs), which are covalent attachment of encoding double stranded DNA to small-molecule created using a combinatio...More data for this Ligand-Target Pair
Affinity DataIC50: <2nMpH: 9.5 T: 2°CAssay Description:Selection of DNA-encoded libraries (DELs), which are covalent attachment of encoding double stranded DNA to small-molecule created using a combinatio...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of topoisomerase I activity was determined in vitro by using the cleavable complex assay(calf thymus)More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 12.4nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human CCR2 in THP1 cells assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Deltagen Research Laboratories (Former Combichem)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]MCP1 from human CCR2b in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of topoisomerase I activity was determined in vitro by using the cleavable complex assay(calf thymus)More data for this Ligand-Target Pair
Affinity DataIC50: 15nMpH: 9.5 T: 2°CAssay Description:Selection of DNA-encoded libraries (DELs), which are covalent attachment of encoding double stranded DNA to small-molecule created using a combinatio...More data for this Ligand-Target Pair