Affinity DataKi: 140nMAssay Description:Displacement of [125I]orexin-A from human OX1R expressed in CHO cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Displacement of [125I]orexin-A from human OX2R expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 411nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 516nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 583nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries
Curated by ChEMBL
Toray Industries
Curated by ChEMBL
Affinity DataIC50: 796nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair