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Found 121 with Last Name = 'nagahara' and Initial = 't'
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]orexin-A from human OX1R expressed in CHO cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataKi:  770nMAssay Description:Displacement of [125I]orexin-A from human OX2R expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146539(2-[4-(6-Chloro-naphthalene-2-sulfonyl)-piperazine-...)
Affinity DataIC50:  7.80nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146534(CHEMBL100732 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146534(CHEMBL100732 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146538(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146536(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  24nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146536(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146532(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146531(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433895(CHEMBL2380435)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433893(CHEMBL2380437)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146537(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  45nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433897(CHEMBL2380433)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146535(CHEMBL99483 | [4-(6-Chloro-naphthalene-2-sulfonyl)...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146535(CHEMBL99483 | [4-(6-Chloro-naphthalene-2-sulfonyl)...)
Affinity DataIC50:  60nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataIC50:  70nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154263(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-isopropyl...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154267(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(4,5,6,7-tet...)
Affinity DataIC50:  83nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433885(CHEMBL2380571)
Affinity DataIC50:  86nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041220(1,2-bis(5-amidinobenzofuran-2-yl)ethane | 2-(2-{5-...)
Affinity DataIC50:  100nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154264(CHEMBL365654 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  105nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433886(CHEMBL2380570)
Affinity DataIC50:  107nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154265(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-ethyl-4,5...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433889(CHEMBL2380567)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433900(CHEMBL2380430)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146540(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433894(CHEMBL2380436)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041218(3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-1-(1...)
Affinity DataIC50:  160nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154270(CHEMBL182957 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154271(CHEMBL185539 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  190nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041221(3-(7-Carbamimidoyl-naphthalen-2-yl)-2-[4-((S)-pyrr...)
Affinity DataIC50:  200nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154266(CHEMBL181749 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  210nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154275(CHEMBL183960 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  270nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041231(3-(7-Carbamimidoyl-naphthalen-2-yl)-2-[4-((S)-pyrr...)
Affinity DataIC50:  310nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154273(CHEMBL365826 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  320nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041219(3-(6-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-1-(1...)
Affinity DataIC50:  360nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433899(CHEMBL2380431)
Affinity DataIC50:  411nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041217(3-(5-Carbamimidoyl-benzofuran-2-yl)-2-{4-[(S)-1-(1...)
Affinity DataIC50:  500nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041224((R)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataIC50:  500nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433898(CHEMBL2380432)
Affinity DataIC50:  516nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154262(CHEMBL185141 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  550nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146534(CHEMBL100732 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  560nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433896(CHEMBL2380434)
Affinity DataIC50:  583nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50154268(CHEMBL363048 | [4-(6-Chloro-naphthalene-2-sulfonyl...)
Affinity DataIC50:  640nMAssay Description:Inhibitory concentration against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041216(2-(2-{4-[(S)-1-(1-Imino-ethyl)-pyrrolidin-3-yloxy]...)
Affinity DataIC50:  640nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146533(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibitory activity of the compound against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50433891(CHEMBL2380565)
Affinity DataIC50:  796nMAssay Description:Antagonist activity at human TRPV1 transfected in CHOK1 cells assessed as inhibition of capsaicin-induced intracellular calcium level measured for 12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146537(4-(6-Chloro-naphthalene-2-sulfonyl)-1-(5-methyl-4,...)
Affinity DataIC50:  820nMAssay Description:In vitro inhibitory activity of the compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50041223(3-(6-Carbamimidoyl-benzofuran-2-yl)-2-{4-[(S)-1-(1...)
Affinity DataIC50:  840nMAssay Description:In vitro evaluation for the concentration needed for inhibiting factor Xa by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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