Compile Data Set for Download or QSAR
maximum 50k data
Found 49 with Last Name = 'nakagawa' and Initial = 'r'
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215149(CHEMBL108634)
Affinity DataIC50:  1.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50147362(CHEMBL330407 | ST-3100)
Affinity DataIC50:  1.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215145(CHEMBL322529)
Affinity DataIC50:  2.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215150(CHEMBL324397)
Affinity DataIC50:  2.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081427((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471733(CHEMBL319183)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471746(CHEMBL422246)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215153(CHEMBL108621)
Affinity DataIC50:  3.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215143(CHEMBL110326)
Affinity DataIC50:  3.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215151(CHEMBL107416)
Affinity DataIC50:  3.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471747(CHEMBL102557)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471741(CHEMBL103333)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50147362(CHEMBL330407 | ST-3100)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  4.00E+3nMAssay Description:The compound was evaluated for the anti-tubulin activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215148(CHEMBL108518)
Affinity DataIC50:  4.00E+3nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471754(CHEMBL103062)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471750(CHEMBL441739)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471736(CHEMBL317013)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471751(CHEMBL103856)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471742(CHEMBL102711)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471745(CHEMBL103329)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471752(CHEMBL102838)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471735(CHEMBL103288)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471749(CHEMBL316750)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471732(CHEMBL102944)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215144(CHEMBL322532)
Affinity DataIC50: >1.00E+4nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471734(CHEMBL103582)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471743(CHEMBL102949)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215146(CHEMBL317022)
Affinity DataIC50: >1.00E+4nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215152(CHEMBL320117)
Affinity DataIC50: >1.00E+4nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50215147(CHEMBL107424)
Affinity DataIC50: >1.00E+4nMAssay Description:Tubulin polymerization inhibitory activity using bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471744(CHEMBL105075)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471740(CHEMBL102702)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471738(CHEMBL322446)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471737(CHEMBL105217)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471753(CHEMBL102235)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471731(CHEMBL320679)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471739(CHEMBL103174)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471755(CHEMBL103653)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50471748(CHEMBL322173)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081428((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081429((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.90E+4nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081429((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081428((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.02E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081426((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.32E+5nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081427((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.72E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081426((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081431(7,16-dihydroxy-5,14-dimethyl-(1S,13S,16R)-2-oxa-14...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081431(7,16-dihydroxy-5,14-dimethyl-(1S,13S,16R)-2-oxa-14...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed