TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:Affinity to mu-receptor, using [3H]DAMGO as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 134nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 237nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetMu-type opioid receptor(GUINEA PIG)
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to mu-receptor, using [3H]DAMGO as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to mu-receptor, using [3H]DAMGO as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to mu-receptor, using [3H]DAMGO as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair