Compile Data Set for Download or QSAR
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Found 230 with Last Name = 'pérez-pérez' and Initial = 'mj'
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116370(1-Benzyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  4nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116384(1-Benzyl-3-cyclopropylmethyl-1H-1,3,4b,9-tetraaza-...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116371(3-Allyl-1-benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  5nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116382(1-Benzyl-3-isobutyl-1H-1,3,4b,9-tetraaza-fluorene-...)
Affinity DataKi:  6.30nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116375(1-(4-Methoxy-benzyl)-3-propyl-1H-1,3,4b,9-tetraaza...)
Affinity DataKi:  8.30nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116368(1-Benzyl-7-methoxy-3-propyl-1H-1,3,4b,9-tetraaza-f...)
Affinity DataKi:  10nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116373(1-Benzyl-3-prop-2-ynyl-1H-1,3,4b,9-tetraaza-fluore...)
Affinity DataKi:  14nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116382(1-Benzyl-3-isobutyl-1H-1,3,4b,9-tetraaza-fluorene-...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116367(1-Benzyl-7-phenyl-3-propyl-1H-1,3,4b,9-tetraaza-fl...)
Affinity DataKi:  35nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116379(1-Benzyl-3-ethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  36nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116371(3-Allyl-1-benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116370(1-Benzyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116377(1-(3-Methyl-benzyl)-3-propyl-1H-1,3,4b,9-tetraaza-...)
Affinity DataKi:  68nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116381(1,3-Dibenzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dio...)
Affinity DataKi:  77nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116375(1-(4-Methoxy-benzyl)-3-propyl-1H-1,3,4b,9-tetraaza...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116373(1-Benzyl-3-prop-2-ynyl-1H-1,3,4b,9-tetraaza-fluore...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116366(1-Benzyl-3-cyclohexylmethyl-1H-1,3,4b,9-tetraaza-f...)
Affinity DataKi:  114nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116370(1-Benzyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116373(1-Benzyl-3-prop-2-ynyl-1H-1,3,4b,9-tetraaza-fluore...)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116371(3-Allyl-1-benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  161nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116368(1-Benzyl-7-methoxy-3-propyl-1H-1,3,4b,9-tetraaza-f...)
Affinity DataKi:  179nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116369(1-Benzyl-7-phenyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  200nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116374(1-Benzyl-7-methoxy-1H-1,3,4b,9-tetraaza-fluorene-2...)
Affinity DataKi:  210nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116380(1-Benzyl-3-(4-methoxy-benzyl)-1H-1,3,4b,9-tetraaza...)
Affinity DataKi:  213nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116384(1-Benzyl-3-cyclopropylmethyl-1H-1,3,4b,9-tetraaza-...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332931(1-[4-(1,1-Dioxo-1H-1lambda-6-naphtho[1,8-cd]isothi...)
Affinity DataKi:  270nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50200995(1-[6-[1,1-(diphenyl)-1-(4-pyridyl)methoxy]hexyl]th...)
Affinity DataKi:  290nMAssay Description:Inhibition of TK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332938(5-Bromo-1-[4-(2,2-dioxo-4,5-dihydro-3H-2lambda-6-t...)
Affinity DataKi:  300nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116379(1-Benzyl-3-ethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116378(1-Benzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dione |...)
Affinity DataKi:  370nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116372(1-Benzyl-7-tert-butyl-3-propyl-1H-1,3,4b,9-tetraaz...)
Affinity DataKi:  385nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332930(5-methyl-1-(4-(2-oxobenzo[cd]indol-1(2H)-yl)but-2-...)
Affinity DataKi:  420nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50118490(1-[(Z)-4-(triphenylmethoxy)-2-butenyl]thymine | 5-...)
Affinity DataKi:  500nMAssay Description:Inhibition of TK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116383(1-Benzyl-7-tert-butyl-1H-1,3,4b,9-tetraaza-fluoren...)
Affinity DataKi:  555nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332937(1-[4-(2,2-Dioxo-4,5-dihydro-3H-2lambda-6-thia-1,2a...)
Affinity DataKi:  570nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116379(1-Benzyl-3-ethyl-1H-1,3,4b,9-tetraaza-fluorene-2,4...)
Affinity DataKi:  584nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332935(CHEMBL1631395 | N-(1-(4-(5-methyl-2,4-dioxo-3,4-di...)
Affinity DataKi:  930nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116372(1-Benzyl-7-tert-butyl-3-propyl-1H-1,3,4b,9-tetraaz...)
Affinity DataKi:  950nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116385(4-(1-Benzyl-2,4-dioxo-1,4-dihydro-2H-1,3,4b,9-tetr...)
Affinity DataKi:  1.13E+3nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332932(5-methyl-1-(4-(2-oxo-2,4,5,6-tetrahydro-1H-imidazo...)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116372(1-Benzyl-7-tert-butyl-3-propyl-1H-1,3,4b,9-tetraaz...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116376(1-Methyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]-DPCPX from CHO cell membrane expressing human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332936(1-(4-(8-amino-2-oxo-2,4,5,6-tetrahydro-1H-imidazo[...)
Affinity DataKi:  2.46E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116376(1-Methyl-3-propyl-1H-1,3,4b,9-tetraaza-fluorene-2,...)
Affinity DataKi:  3.02E+3nMAssay Description:Ability to displace [125I]- AB-MECA from HEK 293 cell membrane expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332929(((2R,3S,5R)-3-hydroxy-5-(5-methyl-2,4-dioxo-3,4-di...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332933(CHEMBL1631396 | N-(1-(4-(5-methyl-2,4-dioxo-3,4-di...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50332934(1-(4-(5-amino-2-oxo-2,4,5,6-tetrahydro-1H-imidazo[...)
Affinity DataKi:  7.07E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis Thymidine monophosphate kinase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)

Curated by ChEMBL
LigandPNGBDBM50116381(1,3-Dibenzyl-1H-1,3,4b,9-tetraaza-fluorene-2,4-dio...)
Affinity DataKi:  2.58E+4nMAssay Description:Displacement of [3H]-ZM-241,385 from CHO cell membrane expressing human Adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50118502(5-Methyl-1-(2-trityloxymethyl-benzyl)-1H-pyrimidin...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with gancicclovirMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50118502(5-Methyl-1-(2-trityloxymethyl-benzyl)-1H-pyrimidin...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with BVAraUMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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