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Found 1884 with Last Name = 'pecchi' and Initial = 's'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.135nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.178nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.209nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.324nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415153(CHEMBL569307)
Affinity DataKi:  0.692nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415144(CHEMBL583051)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415145(CHEMBL571121)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415153(CHEMBL569307)
Affinity DataKi:  1.51nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415153(CHEMBL569307)
Affinity DataKi:  1.55nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415145(CHEMBL571121)
Affinity DataKi:  1.66nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415152(CHEMBL569760)
Affinity DataKi:  2.09nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473413(CHEMBL126487)
Affinity DataKi:  2.30nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415153(CHEMBL569307)
Affinity DataKi:  2.34nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50064609(6-acetoxy-8-azonia-bicyclo[3.2.1]octane | Acetic a...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415145(CHEMBL571121)
Affinity DataKi:  3.31nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM86291(3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxyisox...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415145(CHEMBL571121)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412182(CHEMBL539120)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412177(CHEMBL493979)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415153(CHEMBL569307)
Affinity DataKi:  4.27nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473417(CHEMBL129827)
Affinity DataKi:  4.5nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473417(CHEMBL129827)
Affinity DataKi:  4.5nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415145(CHEMBL571121)
Affinity DataKi:  4.57nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM86291(3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxyisox...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity to human cloned muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415158(CHEMBL569712)
Affinity DataKi:  6.61nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415144(CHEMBL583051)
Affinity DataKi:  6.76nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473414(CHEMBL129790)
Affinity DataKi:  6.80nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473414(CHEMBL129790)
Affinity DataKi:  6.80nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415144(CHEMBL583051)
Affinity DataKi:  7.08nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415152(CHEMBL569760)
Affinity DataKi:  7.24nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415144(CHEMBL583051)
Affinity DataKi:  7.76nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473431(CHEMBL128610)
Affinity DataKi:  8nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415158(CHEMBL569712)
Affinity DataKi:  8.91nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415154(CHEMBL568870)
Affinity DataKi:  9.12nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415154(CHEMBL568870)
Affinity DataKi:  9.33nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50412176(CHEMBL493980)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415152(CHEMBL569760)
Affinity DataKi:  10.2nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50415157(CHEMBL583027)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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