Found 7 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50241132'
Affinity DataKi: 0.135nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M3 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.135nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research
Curated by PDSP Ki Database
National Institute For Medical Research
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research
Curated by PDSP Ki Database
National Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataKi: 0.501nMAssay Description:Binding affinity to Muscarinic acetylcholine receptor M3 by measuring its ability to displace [3H]N-methylscopolamine binding in rat submandibulary g...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Compound was evaluated for its binding affinity at human muscarinic receptor m3 by the displacement of [3H]NMS radioligand using membranes from trans...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research
Curated by PDSP Ki Database
National Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataEC50: 0.0500nMAssay Description:Stimulation of disulfide bond cross-linking formation in rat M3'(3C)-Xa receptor A91C/T549C mutant expressed in african green monkey COS7 cells by sc...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Medical Research
Curated by PDSP Ki Database
National Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataEC50: 0.195nMAssay Description:Stimulation of disulfide bond cross-linking formation in rat M3'(3C)-Xa receptor F92C/F550C mutant expressed in african green monkey COS7 cells by sc...More data for this Ligand-Target Pair