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Found 150 with Last Name = 'petersen' and Initial = 'h'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080399((2R,3R,4S,5R)-2-[6-((1R,2R)-2-Hydroxy-cyclopentyla...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080389((2S,3S,4R,5R)-2-Chloromethyl-5-[2-chloro-6-(4-phen...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080400((2R,3R,4S,5R)-2-[2-Chloro-6-(piperidin-1-ylamino)-...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2A receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080358(1-{2-[2,2-Bis-(2-chloro-phenyl)-vinyloxy]-ethyl}-1...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080367((R)-1-{2-[(Z)-2-(2-Chloro-phenyl)-2-phenyl-vinylox...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080382((R)-1-{2-[(Z)-2-(2-Chloro-phenyl)-2-o-tolyl-vinylo...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080337((R)-1-{2-[2,2-Bis-(3-methyl-thiophen-2-yl)-vinylox...)
Affinity DataKi:  14nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080395((2R,3R,4S,5R)-2-[2-Chloro-6-((S)-1-methyl-2-phenox...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080376((R)-1-{2-[(E)-2-(3-Methyl-thiophen-2-yl)-2-o-tolyl...)
Affinity DataKi:  17nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080335((R)-1-[2-(2,2-Di-o-tolyl-vinyloxy)-ethyl]-piperidi...)
Affinity DataKi:  19nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080327(1-{2-[(Z)-2-(2-Fluoro-phenyl)-2-o-tolyl-vinyloxy]-...)
Affinity DataKi:  19nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080375((R)-1-[2-((E)-2-Phenyl-2-o-tolyl-vinyloxy)-ethyl]-...)
Affinity DataKi:  21nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080390((2R,3R,4S,5R)-2-(6-(2-methyl-benzylamino)-9H-purin...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2A receptor of rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080368(1-[2-(2,2-Di-o-tolyl-vinyloxy)-ethyl]-1,2,5,6-tetr...)
Affinity DataKi:  26nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080388((R)-1-{2-[(E)-2-(3-Fluoro-phenyl)-2-o-tolyl-vinylo...)
Affinity DataKi:  28nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080331((R)-1-{2-[(Z)-2-(4-Fluoro-2-methyl-phenyl)-2-o-tol...)
Affinity DataKi:  30nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080355((R)-1-{2-[2,2-Bis-(2-ethyl-phenyl)-vinyloxy]-ethyl...)
Affinity DataKi:  32nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080365((R)-1-{2-[1-(2,4-Dichloro-phenyl)-1-(3-methyl-thio...)
Affinity DataKi:  32nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080328((R)-1-{2-[Bis-(2-chloro-phenyl)-methyleneaminooxy]...)
Affinity DataKi:  39nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080373((R)-1-{2-[1-(2-Fluoro-phenyl)-1-o-tolyl-meth-(Z)-y...)
Affinity DataKi:  41nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080369((S)-1-{2-[Bis-(3-methyl-thiophen-2-yl)-methyleneam...)
Affinity DataKi:  41nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080397((2R,3R,4S,5R)-2-[2-Chloro-6-(1-methyl-2-phenoxy-et...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080359(1-{2-[2,2-Bis-(2-ethyl-phenyl)-vinyloxy]-ethyl}-1,...)
Affinity DataKi:  47nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080344(1-(2-Benzhydrylideneaminooxy-ethyl)-1,2,5,6-tetrah...)
Affinity DataKi:  47nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080370((R)-1-{2-[(Z)-2-(3-Fluoro-phenyl)-2-o-tolyl-vinylo...)
Affinity DataKi:  48nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080323((R)-1-[2-((Z)-2-Phenyl-2-o-tolyl-vinyloxy)-ethyl]-...)
Affinity DataKi:  49nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080333((R)-1-{2-[(E)-2-(2,4-Difluoro-phenyl)-2-(2,5-diflu...)
Affinity DataKi:  51nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080330((R)-1-{2-[(E)-2-(2-Chloro-phenyl)-2-phenyl-vinylox...)
Affinity DataKi:  52nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080340((R)-1-{2-[(2,4-Difluoro-phenyl)-(2,5-difluoro-phen...)
Affinity DataKi:  52nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080336((R)-1-{2-[2,2-Bis-(2-chloro-phenyl)-vinyloxy]-ethy...)
Affinity DataKi:  52nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080324(1-(2-Di-o-tolylmethyleneaminooxy-ethyl)-1,2,5,6-te...)
Affinity DataKi:  55nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080387((R)-1-{2-[1-(1-Methyl-1H-pyrrol-2-yl)-1-phenyl-met...)
Affinity DataKi:  59nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080374((R)-1-{2-[2,2-Bis-(4-fluoro-2-methyl-phenyl)-vinyl...)
Affinity DataKi:  61nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080341(1-{2-[(Z)-2-(3-Chloro-phenyl)-2-o-tolyl-vinyloxy]-...)
Affinity DataKi:  64nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080381((R)-1-{2-[2,2-Bis-(2-chloro-4-fluoro-phenyl)-vinyl...)
Affinity DataKi:  66nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50368628(ABT-569 | Abbott-70569 | Abbott-70569.1 | Gabitril...)
Affinity DataKi:  67nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080354((R)-1-{2-[1-(3-Methyl-thiophen-2-yl)-1-o-tolyl-met...)
Affinity DataKi:  70nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080354((R)-1-{2-[1-(3-Methyl-thiophen-2-yl)-1-o-tolyl-met...)
Affinity DataKi:  70nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080364((R)-1-(2-Di-o-tolylmethyleneaminooxy-ethyl)-piperi...)
Affinity DataKi:  71nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080334((R)-1-{2-[1-(3-Methyl-thiophen-2-yl)-1-thiophen-2-...)
Affinity DataKi:  74nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080396((2R,3R,4R,5R)-5-(6-Cyclohexylamino-purin-9-yl)-2-h...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080380(1-{2-[2,2-Bis-(4-fluoro-2-methyl-phenyl)-vinyloxy]...)
Affinity DataKi:  79nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080346((R)-1-(2-Benzhydrylideneaminooxy-ethyl)-piperidine...)
Affinity DataKi:  81nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080369((S)-1-{2-[Bis-(3-methyl-thiophen-2-yl)-methyleneam...)
Affinity DataKi:  82nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080350((S)-1-{2-[1-(3-Methyl-thiophen-2-yl)-1-o-tolyl-met...)
Affinity DataKi:  83nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080332((R)-1-{2-[(E)-2-(3-Methoxy-phenyl)-2-o-tolyl-vinyl...)
Affinity DataKi:  83nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080379((R)-1-[2-(2,2-Diphenyl-vinyloxy)-ethyl]-piperidine...)
Affinity DataKi:  86nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080384((R)-1-{2-[1-(3-Methoxy-phenyl)-1-(3-methyl-thiophe...)
Affinity DataKi:  87nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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