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Found 19 with Last Name = 'ravaschino' and Initial = 'e'
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM25298((1-hydroxy-1-phosphonoheptyl)phosphonic acid | CHE...)
Affinity DataKi:  400nMAssay Description:Inhibition of trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173056((1-Amino-1-phosphono-hexyl)-phosphonic acid | CHEM...)
Affinity DataIC50:  382nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM25298((1-hydroxy-1-phosphonoheptyl)phosphonic acid | CHE...)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117543(2-Amino-4-{3-methyl-1-[2-oxo-2-(toluene-4-sulfonyl...)
Affinity DataIC50:  2.00E+3nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173058((1-Amino-1-phosphono-heptyl)-phosphonic acid | CHE...)
Affinity DataIC50:  3.57E+3nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173055((1-Amino-1-phosphono-pentyl)-phosphonic acid | CHE...)
Affinity DataIC50:  3.91E+3nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataIC50:  1.72E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173053((1-Amino-1-phosphono-butyl)-phosphonic acid | CHEM...)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173054((1-Amino-1-phosphono-ethyl)-phosphonic acid | CHEM...)
Affinity DataIC50:  6.67E+4nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117545(2-Amino-4-{3-methyl-1-[(1H-tetrazol-5-ylmethyl)-ca...)
Affinity DataIC50:  1.38E+5nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50173057((1-Amino-1-phosphono-propyl)-phosphonic acid | CHE...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibitory concentration against trypanosoma cruzi farnesyl pyrophosphate synthase (TcFPPS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed