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Found 84 with Last Name = 'roberts' and Initial = 'sm'
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070866((2R,3R,4S,5R)-2-[2-Chloro-6-(3-iodo-benzylamino)-p...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070867((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  20nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070864((2R,3R,4S,5S)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  26nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027680(CHEMBL3357975)
Affinity DataKi:  27nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070865((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  31nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070863((2S,3S,4R,5R)-5-(6-Benzylamino-purin-9-yl)-3,4-dih...)
Affinity DataKi:  41nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  54nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  56nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070864((2R,3R,4S,5S)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  74nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070865((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  620nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027677(CHEMBL3344387)
Affinity DataKi:  631nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070867((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027681(CHEMBL3357976)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070866((2R,3R,4S,5R)-2-[2-Chloro-6-(3-iodo-benzylamino)-p...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070866((2R,3R,4S,5R)-2-[2-Chloro-6-(3-iodo-benzylamino)-p...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070863((2S,3S,4R,5R)-5-(6-Benzylamino-purin-9-yl)-3,4-dih...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070863((2S,3S,4R,5R)-5-(6-Benzylamino-purin-9-yl)-3,4-dih...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070864((2R,3R,4S,5S)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi:  4.65E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027679(CHEMBL3344389)
Affinity DataKi:  4.91E+3nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070867((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50070865((2R,3R,4S,5R)-2-(2-Chloro-6-methoxyamino-purin-9-y...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027678(CHEMBL3344388)
Affinity DataKi:  1.09E+4nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027676(CHEMBL3344386)
Affinity DataKi:  2.85E+4nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341705(CHEMBL1766652 | rac-1-[2-(Carboxy)-4-(triphenylmet...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341704(CHEMBL1766653 | rac-1-[2-(Acetamide)-4-(triphenylm...)
Affinity DataKi:  9.80E+4nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341701(CHEMBL1766637 | rac-1-[2-(tert-Butyldiphenylsilylo...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341709(CHEMBL1766648 | rac-1-[2-(Ethylamido)-4-(tert-buty...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341702(CHEMBL1766636 | rac-1-(2-Dimethylamido-4-trityloxy...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341692(CHEMBL1766646 | rac-1-[2-(Acetamide)-4-(tert-butyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341703(CHEMBL1766635 | rac-1-(2-Amido-4-trityloxybutyl)ur...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341693(CHEMBL1766645 | rac-1-[2-(Carboxy)-4-(tert-butyldi...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341695(CHEMBL1766643 | rac-1-[2-(Hydroxyethylamido)-4-tri...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341697(CHEMBL1766641 | rac-1-[2-(Methoxyethylamido)-4-tri...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341706(CHEMBL1766651 | rac-benzyl 2-((2,4-dioxo-3,4-dihyd...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341698(CHEMBL1766640 | rac-1-(2-Morpholinamido-4-tritylox...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341707(CHEMBL1766650 | rac-benzyl 4-(4-(tert-butyldipheny...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341699(CHEMBL1766639 | rac-1-[2-(N,N-Dimethylaminoethylam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341708(CHEMBL1766649 | rac-1-[2-(Diethylamido)-4-(tert-bu...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341700(CHEMBL1766638 | rac-1-[2-(Carboethoxyethylamido)-4...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341696(CHEMBL1766642 | rac-1-[2-(N-Methylpiperazine)amido...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341694(CHEMBL1766644 | rac-1-[2-(Carboxyethylamido)-4-tri...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50341710(CHEMBL1766647 | rac-1-[2-(Methylamido)-4-(tert-but...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dUTPase by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539993(CHEMBL4647500)
Affinity DataIC50:  180nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539980(CHEMBL4644304)
Affinity DataIC50:  550nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539992(CHEMBL4632916)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50027677(CHEMBL3344387)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human NMT1 using GSNKSKPKDASQRRR-NH2 as substrate by CPM fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539975(CHEMBL4633418)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539991(CHEMBL4632704)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50539990(CHEMBL4647034)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human NMT1 using p60 SRC(2 to 16) as substrate by CPM dye based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
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