Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute
Curated by ChEMBL
Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute
Curated by ChEMBL
Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.643nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to insulin receptor by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to IGF1R by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human plasma carboxypeptidase NMore data for this Ligand-Target Pair
Affinity DataKi: 2.17nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to insulin receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from guinea pig tracheaMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase D(Homo sapiens (Human))
University Of Kansas
Curated by ChEMBL
University Of Kansas
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Binding affinity to human recombinant cyclophilin D by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute
Curated by ChEMBL
Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibitory effect on plasmin in bovine plasmaMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 4.97nMAssay Description:Inhibitory effect on Coagulation factor Xa (FXa) from bovine plasmaMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity to IGF1R by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from human expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute
Curated by ChEMBL
Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of bovine pancreatic carboxypeptidase AMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute
Curated by ChEMBL
Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Glaxo Wellcome Medicines Research Centre
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair